SCHEMBL6201668

SCHEMBL6201668

CN(CCO)C(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)(C)S

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSK P43235 12/20 0.40
CA1 P00915 2/20 0.38
CA7 P43166 2/20 0.38
CA2 P00918 1/20 0.38
TDP1 Q9NUW8 1/20 0.36
CYP2D6 P10635 1/20 0.35
CTSS P25774 3/20 0.33
CA12 O43570 1/20 0.33
CA14 Q9ULX7 1/20 0.33
KMT2A Q03164 1/20 0.32
CTSL P07711 1/20 0.32
CTSB P07858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6201666 1.00 CTSK (0.40) CTSKCA1CA7CA2TDP1
SCHEMBL6201206 0.73 CA1 (0.43) CTSKCA1CA7CA2CYP2D6
SCHEMBL3151434 0.73 CA1 (0.43) CTSKCA1CA7CA2CYP2D6
SCHEMBL6202245 0.73 CA1 (0.43) CTSKCA1CA7CA2CYP2D6
SCHEMBL18793620 0.72 CA12 (0.42) CTSKCA1CA7CA2CYP2D6
SCHEMBL31269564 0.71 CTSK (0.44) CTSKCA1CA7CA2CTSS
SCHEMBL13050499 0.70 ACE (0.58) CTSKCTSSCTSLCTSB
SCHEMBL13080563 0.70 ACE (0.58) CTSKCTSSCTSLCTSB
SCHEMBL7897117 0.70 CA1 (0.41) CTSKCA1CA7CA2CYP2D6
SCHEMBL12866689 0.68 CA1 (0.46) CTSKCA1CA7CA2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165532-B1 ANTIBACTERIAL AGENTS VERNALIS OXFORD LTD (GB) 2005-01-12 EP disclosed
US-6503897-B1 N-Formylhydroxylamine derivatives; veterinary medicine; grampositive and gramnegative bacteria BRITISH BIOTECH PHARMACEUTICALS LTD. (GB) 2003-01-07 US disclosed