SCHEMBL6202261

SCHEMBL6202261

O=C(NCc1ccc(Cl)cc1)c1cnc2c(S(=O)(=O)NCCN(CCO)CCO)cc(F)cc2c1O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.41
EGLN1 Q9GZT9 1/20 0.38
CXCR4 P61073 1/20 0.37
NR3C1 P04150 1/20 0.37
LMNA P02545 1/20 0.37
TUBB P07437 2/20 0.36
TP53 P04637 1/20 0.35
PTGER4 P35408 1/20 0.35
PTGER2 P43116 1/20 0.35
CYP1A2 P05177 2/20 0.35
HPGD P15428 2/20 0.35
CYP2C19 P33261 2/20 0.35
CCKBR P32239 1/20 0.35
CYP2C9 P11712 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
POLA1 P09884 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
ALDH1A1 P00352 1/20 0.34
CNR2 P34972 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6199253 0.92 MCL1 (0.44) MCL1EGLN1CXCR4NR3C1LMNA
SCHEMBL6202413 0.91 MCL1 (0.43) MCL1EGLN1CXCR4NR3C1LMNA
SCHEMBL6201234 0.89 MCL1 (0.42) MCL1EGLN1CXCR4NR3C1LMNA
SCHEMBL6201656 0.88 MCL1 (0.44) MCL1EGLN1CXCR4NR3C1LMNA
SCHEMBL6199074 0.88 MCL1 (0.44) MCL1EGLN1CXCR4NR3C1LMNA
SCHEMBL6201979 0.88 MCL1 (0.52) MCL1EGLN1CXCR4NR3C1LMNA
SCHEMBL6197440 0.88 MCL1 (0.41) MCL1EGLN1CXCR4NR3C1LMNA
SCHEMBL6200365 0.87 EGLN1 (0.42) MCL1EGLN1NR3C1LMNATUBB
SCHEMBL6199403 0.87 TUBB (0.40) MCL1EGLN1CXCR4NR3C1LMNA
SCHEMBL6200751 0.87 MCL1 (0.41) MCL1EGLN1CXCR4NR3C1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042295-B1 4-HYDROXYQUINOLINE-3-CARBOXAMIDES AND HYDRAZIDES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN CO LLC (US) 2005-09-07 EP claimed