SCHEMBL6202476

SCHEMBL6202476

CN(C)CCOc1ccc2[nH]c3c(c2c1)C(=O)c1cc2c(cc1-3)OCCO2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.46
TOP2A P11388 2/20 0.43
ESR1 P03372 2/20 0.39
KDR P35968 2/20 0.39
BCHE P06276 2/20 0.39
MAOA P21397 2/20 0.39
ACHE P22303 2/20 0.39
MAOB P27338 2/20 0.39
TNKS O95271 2/20 0.39
ALK Q9UM73 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
NUAK1 O60285 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
PDGFRB P09619 1/20 0.38
PDGFRA P16234 1/20 0.38
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7236878 0.99 PARP1 (0.46) PARP1TOP2AESR1KDRBCHE
SCHEMBL6203062 0.84 PARP1 (0.46) PARP1TOP2AESR1KDRTNKS
Hydrochloric Acid SCHEMBL7235812 0.83 PARP1 (0.45) PARP1TOP2AESR1KDRTNKS
SCHEMBL6202601 0.83 KDM4E (0.47) PARP1TOP2AESR1KDRTNKS
SCHEMBL6197999 0.83 TOP2A (0.54) PARP1TOP2AESR1TNKSALK
Hydrochloric Acid SCHEMBL7236341 0.82 KDM4E (0.46) PARP1TOP2AESR1KDRTNKS
Hydrochloric Acid SCHEMBL7236484 0.82 TOP2A (0.53) PARP1TOP2AESR1TNKSALK
Hydrochloric Acid SCHEMBL7227302 0.78 PARP1 (0.35) PARP1TOP2AESR1MAOAMAOB
Hydrochloric Acid SCHEMBL7227308 0.78 PARP1 (0.35) PARP1TOP2AESR1MAOAMAOB
SCHEMBL6203316 0.74 PARP1 (0.47) PARP1TOP2AESR1KDRMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1266887-B1 Indenoindoline derivatives, their process of preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2005-08-17 EP disclosed
EP-1266887-A2 Indenoindoline derivatives, their process of preparation and pharmaceutical compositions containing them Les Laboratoires Servier (FR) 2002-12-18 EP disclosed