SCHEMBL6202557

SCHEMBL6202557

O=C(Cc1cccnn1)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 1/20 0.51
CYP1A2 P05177 3/20 0.50
CTDSP1 Q9GZU7 1/20 0.50
RAB9A P51151 2/20 0.49
NPC1 O15118 1/20 0.49
PLOD2 O00469 2/20 0.46
HPGD P15428 3/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2C19 P33261 2/20 0.46
CYP2C9 P11712 2/20 0.46
ALDH1A1 P00352 2/20 0.46
HIF1A Q16665 2/20 0.46
PLOD3 O60568 1/20 0.46
CYP2D6 P10635 1/20 0.46
PLOD1 Q02809 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.45
KDM4E B2RXH2 2/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
MAPK1 P28482 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11318815 0.81 CYP1A2 (0.56) VNN1CYP1A2CTDSP1CYP2C9KDM4E
Hydrochloric Acid SCHEMBL27803205 0.79 CYP1A2 (0.54) VNN1CYP1A2CTDSP1CYP2C9KDM4E
SCHEMBL2051943 0.78 RAB9A (0.75) CYP1A2RAB9ANPC1PLOD2HPGD
SCHEMBL6011931 0.78 RAB9A (0.75) CYP1A2RAB9ANPC1PLOD2HPGD
SCHEMBL11636011 0.77 KDM4E (0.55) CYP1A2RAB9ANPC1PLOD2HPGD
SCHEMBL29017606 0.76 RAB9A (0.73) CYP1A2RAB9ANPC1PLOD2HPGD
SCHEMBL30333799 0.76 RAB9A (0.73) CYP1A2RAB9ANPC1PLOD2HPGD
SCHEMBL29986829 0.76 RAB9A (0.73) CYP1A2RAB9ANPC1PLOD2HPGD
Hydrochloric Acid SCHEMBL11622188 0.76 RAB9A (0.73) CYP1A2RAB9ANPC1PLOD2HPGD
Bromide SCHEMBL28156394 0.76 RAB9A (0.73) CYP1A2RAB9ANPC1PLOD2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050272036-A1 Ketones ASTRAZENECA AB (SE) 2005-12-08 US disclosed
CN-1681763-A Chemical compounds ASTRAZENECA AB (SE) 2005-10-12 CN disclosed
EP-1549600-A1 KETONES AstraZeneca AB (SE) 2005-07-06 EP disclosed
WO-2004011410-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2004-02-05 WO disclosed
EP-0715624-B1 PROCESS FOR THE PREPARATION OF BENZODIAZEPINE COMPOUNDS USEFUL AS ANTAGONISTS OF CCK OR OF GASTRINE YAMANOUCHI PHARMA CO LTD (JP) 1998-04-08 EP disclosed
US-5728829-A MULTISTAGE REACTION OF N-PROTECTED BENZOTRIAZOLYL GLYCINE DERIVATIVE WITH AMINOKETONE, THEN REACTION WITH AMMONIA AND ACID CATALYZED CYCLIZATION FERRING-RESEARCH LIMITED (GB) 1998-03-17 US disclosed
EP-0715624-A1 PROCESS FOR THE PREPARATION OF BENZODIAZEPINE COMPOUNDS USEFUL AS ANTAGONISTS OF CCK OR OF GASTRINE YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1996-06-12 EP disclosed
WO-1995006040-A1 BENZODIAZEPINE COMPOUNDS USEFUL AS ANTAGONISTS OF CCK OR OF GASTRINE YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1995-03-02 WO disclosed