SCHEMBL6202735

SCHEMBL6202735

COc1cccc(CNc2nc(N(CCO)C(C)C)nc3c2N(C(C)C)NN3C(C)C)c1O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNE1 P24864 5/20 0.44
CDK2 P24941 5/20 0.44
PKM P14618 4/20 0.43
GAA P10253 9/20 0.41
NPC1 O15118 5/20 0.41
RAB9A P51151 4/20 0.41
ALOX5 P09917 1/20 0.41
CCNT1 O60563 2/20 0.39
CCNT2 O60583 2/20 0.39
CCNE2 O96020 2/20 0.39
CDK9 P50750 2/20 0.39
ALDH1A1 P00352 6/20 0.39
MAPT P10636 5/20 0.39
ALOX12 P18054 3/20 0.39
NPSR1 Q6W5P4 1/20 0.39
GFER P55789 1/20 0.39
TSHR P16473 1/20 0.38
HPGD P15428 3/20 0.38
HTT P42858 2/20 0.38
MEN1 O00255 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6205419 0.92 CCNE1 (0.36) CCNE1CDK2PKMGAANPC1
SCHEMBL6204991 0.86 PKM (0.42) CCNE1CDK2PKMGAANPC1
SCHEMBL6203391 0.83 CCNE2 (0.31) CCNE1CDK2CCNT1CCNE2CDK9
SCHEMBL6201113 0.81 CDK1 (0.46) CCNE1CDK2NPC1CCNT1CCNE2
SCHEMBL3444561 0.80 CDK2 (0.50) CCNE1CDK2PKMGAANPC1
SCHEMBL6203896 0.80 CCNE2 (0.37) CCNE1CDK2CCNT1CCNE2CDK9
SCHEMBL3446101 0.79 PKM (0.46) CCNE1CDK2PKMGAANPC1
SCHEMBL3444999 0.78 PKM (0.45) CCNE1CDK2PKMGAANPC1
SCHEMBL3445452 0.78 CDK2 (0.64) CCNE1CDK2PKMGAANPC1
SCHEMBL6205622 0.78 CCNE2 (0.35) CCNE1CDK2CCNT1CCNE2CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP claimed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO claimed