Bicarbonate

Bicarbonate

SCHEMBL6203741

CCOC(=O)c1ccc(N2CCCCC2)s1.CCOC(=O)c1ccc(N2CCCCC2)s1.O=C([O-])[O-].[Cs+].[Cs+]

nearest known ligand 0.45

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.45
HDAC4 P56524 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
LMNA P02545 2/20 0.41
ALDH1A1 P00352 10/20 0.40
MAPT P10636 5/20 0.40
KMT2A Q03164 4/20 0.40
NPC1 O15118 4/20 0.40
RAB9A P51151 4/20 0.40
TSHR P16473 3/20 0.40
PSMD14 O00487 1/20 0.40
PKM P14618 1/20 0.40
KDM4E B2RXH2 4/20 0.40
HPGD P15428 3/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
GAA P10253 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
MEN1 O00255 2/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5224398 0.95 HDAC3 (0.49) HDAC3HDAC4HDAC1HDAC6LMNA
SCHEMBL5227048 0.93 HDAC3 (0.50) HDAC3HDAC4HDAC1HDAC6LMNA
SCHEMBL63716 0.83 HDAC3 (0.44) HDAC3HDAC4HDAC1HDAC6ALDH1A1
SCHEMBL64634 0.82 HDAC3 (0.48) HDAC3HDAC4HDAC1HDAC6LMNA
SCHEMBL64328 0.82 HDAC3 (0.43) HDAC3HDAC4HDAC1HDAC6LMNA
SCHEMBL19579546 0.81 HDAC3 (0.47) HDAC3HDAC4HDAC1HDAC6ALDH1A1
SCHEMBL63685 0.81 KDM4E (0.47) HDAC3HDAC4HDAC1HDAC6LMNA
SCHEMBL21273299 0.81 MAPT (0.43) LMNAALDH1A1MAPTKMT2ANPC1
SCHEMBL3121764 0.81 ALDH1A1 (0.57) HDAC3HDAC4HDAC1HDAC6LMNA
SCHEMBL23630400 0.80 HDAC3 (0.46) HDAC3HDAC4HDAC1HDAC6LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501508-A1 INHIBITORS OF HISTONE DEACETYLASE Astrazeneca AB (SE) 2005-02-02 EP disclosed
WO-2003092686-A1 INHIBITORS OF HISTONE DEACETYLASE ASTRAZENECA AB (SE) 2003-11-13 WO disclosed