SCHEMBL6203933

SCHEMBL6203933

N#CC(CC(=O)c1ccc(Cl)cc1)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.56
MAPT P10636 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
POLB P06746 2/20 0.49
KMT2A Q03164 3/20 0.48
MEN1 O00255 1/20 0.48
MMP2 P08253 3/20 0.46
MMP3 P08254 3/20 0.46
MMP9 P14780 3/20 0.46
MMP13 P45452 2/20 0.46
MMP1 P03956 1/20 0.46
MMP8 P22894 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
GAA P10253 2/20 0.46
KDM4E B2RXH2 1/20 0.46
HSD11B1 P28845 1/20 0.45
CES2 O00748 1/20 0.44
CES1 P23141 1/20 0.44
GSK3B P49841 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6203114 0.94 KMT2A (0.50) PDPK1MAPTL3MBTL1POLBKMT2A
SCHEMBL31326025 0.89 TSHR (0.53) PDPK1MAPTL3MBTL1KMT2AMEN1
SCHEMBL1754734 0.89 TSHR (0.53) PDPK1MAPTL3MBTL1KMT2AMEN1
SCHEMBL27973291 0.85 POLB (0.63) MAPTL3MBTL1POLBKMT2AMEN1
SCHEMBL28727127 0.85 POLB (0.63) MAPTL3MBTL1POLBKMT2AMEN1
SCHEMBL6223072 0.84 ALDH1A1 (0.48) PDPK1MAPTL3MBTL1KMT2AMEN1
SCHEMBL8696883 0.84 KMT2A (0.60) PDPK1MAPTL3MBTL1KMT2AMEN1
SCHEMBL8694320 0.84 KMT2A (0.53) PDPK1MAPTPOLBKMT2AMEN1
SCHEMBL29624410 0.84 KMT2A (0.66) PDPK1POLBKMT2AMEN1KDM4E
SCHEMBL28727237 0.84 KMT2A (0.66) PDPK1POLBKMT2AMEN1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104030870-B A kind of preparation method of beta-cyano ketone NORTHWEST NORMAL UNIVERSITY (CN) 2015-10-28 CN disclosed
CN-104030870-A Method for preparing beta-cyan ketone UNIV NORTHWEST NORMAL 2014-09-10 CN disclosed
US-20050272036-A1 Ketones ASTRAZENECA AB (SE) 2005-12-08 US disclosed
EP-1549600-A1 KETONES AstraZeneca AB (SE) 2005-07-06 EP disclosed
WO-2004011410-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2004-02-05 WO disclosed
US-5753642-A AGRICULTURE, MEDICINE ROHM AND HAAS COMPANY (US) 1998-05-19 US disclosed
CN-1038249-C Dihydropyridazinones, pyridazinones and related compounds as fungicides ROHM & HAAS (US) 1998-05-06 CN disclosed
US-5728694-A Dihydropyridazinones, pyridazinones and related compounds as fungicides ROHM AND HAAS COMPANY (US) 1998-03-17 US disclosed
US-5728715-A FOR MAMMALS, AGRICULTURE, RICE, WHEAT, TOMATOES ROHM AND HAAS COMPANY (US) 1998-03-17 US disclosed
US-5728698-A AGRICULTURAL USE, RICE, WHEAT ROHM AND HAAS COMPANY (US) 1998-03-17 US disclosed
US-5726176-A FOR CONTROLLING AGRICULTURAL AND MAMMALIAN FUNGAL DISEASES ROHM AND HAAS COMPANY (US) 1998-03-10 US disclosed
US-5726162-A FOR CONTROLLING AGRICULTURAL AND MAMMALIAN FUNGAL DISEASES ROHM AND HAAS COMPANY (US) 1998-03-10 US disclosed
US-5631254-A RICE; HUMAN INFECTIONS ROHM AND HAAS COMPANY (US) 1997-05-20 US disclosed
US-5552409-A PHYTOPATHOGENIC, RICE ROHM AND HAAS COMPANY (US) 1996-09-03 US disclosed
EP-0478195-A1 Dihydropyridazinones, pyridazinones and related compounds as fungicides ROHM AND HAAS COMPANY (US) 1992-04-01 EP disclosed