SCHEMBL6204733

SCHEMBL6204733

O=C(NCc1ccc(Cn2ccnc2)cc1)c1c[nH]c2ccc(Cl)cc2c1=O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SNCA P37840 1/20 0.62
NHERF1 O14745 1/20 0.58
TBXAS1 P24557 1/20 0.55
ADORA2A P29274 2/20 0.49
ADORA1 P30542 2/20 0.49
WDR5 P61964 2/20 0.49
GABRP O00591 3/20 0.48
GABRD O14764 3/20 0.48
GABRA1 P14867 3/20 0.48
GABRB1 P18505 3/20 0.48
GABRG2 P18507 3/20 0.48
GABRB3 P28472 3/20 0.48
GABRA5 P31644 3/20 0.48
GABRA3 P34903 3/20 0.48
GABRA2 P47869 3/20 0.48
GABRB2 P47870 3/20 0.48
GABRA4 P48169 3/20 0.48
GABRE P78334 3/20 0.48
GABRA6 Q16445 3/20 0.48
GABRG1 Q8N1C3 3/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6206094 0.93 SNCA (0.56) SNCANHERF1TBXAS1WDR5GABRP
SCHEMBL6205541 0.88 MEN1 (0.52) SNCATBXAS1ADORA2AADORA1POLB
SCHEMBL6204863 0.86 POLB (0.68) SNCAPOLBMAPTTDP1TP53
SCHEMBL6207242 0.82 ADORA2A (0.47) SNCAADORA2AADORA1WDR5
SCHEMBL6204128 0.81 NHERF1 (0.68) SNCANHERF1ADORA2AADORA1GABRP
SCHEMBL6230550 0.81 NHERF1 (0.68) NHERF1ADORA2AADORA1GABRPGABRD
Hydrochloric Acid SCHEMBL6206076 0.80 NHERF1 (0.67) NHERF1ADORA2AADORA1GABRPGABRD
SCHEMBL6205349 0.79 NHERF1 (0.65) NHERF1ADORA2AADORA1GABRPGABRD
SCHEMBL6204032 0.79 POLB (0.68) POLBMAPTTDP1TP53SMN1; SMN2
SCHEMBL6204818 0.78 NHERF1 (0.59) NHERF1ADORA2AADORA1GABRPGABRD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177177-B1 SUBSTITUTED 4-OXO-QUINOLINE-3-CARBOXAMIDES: GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORP (US) 2005-02-23 EP claimed
US-6413956-B1 AGONISTS, ANTAGONISTS OR INVERSE AGONISTS AND LOCALIZATION PROBES FOR GAMMA AMINOBUTYRIC ACID BRAIN RECEPTORS; ANXIETY, DEPRESSION, DOWN SYNDROME, SLEEP AND SEIZURE DISORDERS, OVERDOSE WITH BENZODIAZEPINE DRUGS AND MEMORY ENHANCEMENT NEUROGEN CORPORATION 2002-07-02 US claimed
EP-1177177-B1 SUBSTITUTED 4-OXO-QUINOLINE-3-CARBOXAMIDES: GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORP (US) 2005-02-23 EP disclosed
US-6413956-B1 AGONISTS, ANTAGONISTS OR INVERSE AGONISTS AND LOCALIZATION PROBES FOR GAMMA AMINOBUTYRIC ACID BRAIN RECEPTORS; ANXIETY, DEPRESSION, DOWN SYNDROME, SLEEP AND SEIZURE DISORDERS, OVERDOSE WITH BENZODIAZEPINE DRUGS AND MEMORY ENHANCEMENT NEUROGEN CORPORATION 2002-07-02 US disclosed