SCHEMBL6204772

SCHEMBL6204772

CCOc1cccc2c(=O)c(C(=O)NCCCOC(C)C)c[nH]c12

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.62
MEN1 O00255 5/20 0.61
KMT2A Q03164 5/20 0.61
HPGD P15428 4/20 0.51
MAPT P10636 2/20 0.51
HSD17B10 Q99714 2/20 0.51
L3MBTL1 Q9Y468 2/20 0.51
GAA P10253 1/20 0.51
KDM4E B2RXH2 3/20 0.50
CNR1 P21554 1/20 0.50
CNR2 P34972 1/20 0.50
POLB P06746 3/20 0.49
TDP1 Q9NUW8 1/20 0.49
RAB9A P51151 3/20 0.48
NPC1 O15118 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6204607 0.90 ALDH1A1 (0.75) ALDH1A1MEN1KMT2AHPGDMAPT
SCHEMBL6206536 0.89 ALDH1A1 (0.77) ALDH1A1MEN1KMT2AHPGDMAPT
SCHEMBL6204974 0.79 POLB (0.64) ALDH1A1MEN1KMT2AHPGDMAPT
SCHEMBL6204768 0.78 KDM4E (0.80) ALDH1A1MEN1KMT2AHPGDMAPT
SCHEMBL6205058 0.78 POLB (0.62) ALDH1A1MEN1KMT2AHPGDMAPT
SCHEMBL17424065 0.77 CNR2 (0.60) ALDH1A1MEN1KMT2AHPGDMAPT
SCHEMBL17424082 0.76 ALDH1A1 (0.61) ALDH1A1MEN1KMT2AHPGDMAPT
SCHEMBL2971885 0.76 ALDH1A1 (0.73) ALDH1A1MEN1KMT2AHPGDMAPT
SCHEMBL6206717 0.75 POLB (0.54) ALDH1A1MEN1KMT2AHPGDMAPT
SCHEMBL6205750 0.75 ALDH1A1 (0.81) ALDH1A1MEN1KMT2AHPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177177-B1 SUBSTITUTED 4-OXO-QUINOLINE-3-CARBOXAMIDES: GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORP (US) 2005-02-23 EP claimed