SCHEMBL6204849

SCHEMBL6204849

O=C(NCc1ccc(CN2CCOCC2)cc1)c1c[nH]c2ccccc2c1=O

nearest known ligand 0.64

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 6/20 0.60
ALDH1A1 P00352 2/20 0.59
POLB P06746 1/20 0.58
MAPT P10636 1/20 0.58
NPC1 O15118 1/20 0.55
RAB9A P51151 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
F2 P00734 1/20 0.52
HSD17B10 Q99714 1/20 0.52
HDAC1 Q13547 1/20 0.51
HDAC6 Q9UBN7 1/20 0.51
HPGD P15428 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6205556 0.99 HRH3 (0.59) HRH3ALDH1A1POLBMAPTNPC1
SCHEMBL6205238 0.91 NPC1 (0.55) HRH3ALDH1A1POLBMAPTNPC1
Hydrochloric Acid SCHEMBL6206718 0.90 NPC1 (0.54) HRH3ALDH1A1POLBMAPTNPC1
SCHEMBL6205197 0.88 POLB (0.61) ALDH1A1POLBMAPTNPC1RAB9A
SCHEMBL6206000 0.88 HRH3 (0.53) HRH3ALDH1A1POLBMAPTNPC1
Hydrochloric Acid SCHEMBL6208393 0.87 HRH3 (0.53) HRH3ALDH1A1POLBMAPTNPC1
SCHEMBL6983693 0.86 HPGD (0.55) ALDH1A1POLBMAPTNPC1RAB9A
SCHEMBL6206009 0.85 HPGD (0.58) HRH3ALDH1A1POLBMAPTNPC1
SCHEMBL6204682 0.85 TSHR (0.61) ALDH1A1POLBMAPTF2HSD17B10
Hydrochloric Acid SCHEMBL6206697 0.84 TSHR (0.60) ALDH1A1POLBMAPTF2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177177-B1 SUBSTITUTED 4-OXO-QUINOLINE-3-CARBOXAMIDES: GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORP (US) 2005-02-23 EP claimed
US-6413956-B1 AGONISTS, ANTAGONISTS OR INVERSE AGONISTS AND LOCALIZATION PROBES FOR GAMMA AMINOBUTYRIC ACID BRAIN RECEPTORS; ANXIETY, DEPRESSION, DOWN SYNDROME, SLEEP AND SEIZURE DISORDERS, OVERDOSE WITH BENZODIAZEPINE DRUGS AND MEMORY ENHANCEMENT NEUROGEN CORPORATION 2002-07-02 US claimed