SCHEMBL6205553

SCHEMBL6205553

CC(C)(C)OC(=O)Nc1ccccc1NC(=O)c1ccc(N2CCNCC2)nc1.Nc1ccccc1NC(=O)c1ccc(N2CCNCC2)nc1

nearest known ligand 0.64

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 14/20 0.64
KCNH2 Q12809 4/20 0.61
HDAC2 Q92769 7/20 0.59
HDAC3 O15379 5/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5225414 0.94 KCNH2 (0.57) HDAC1KCNH2HDAC2HDAC3
SCHEMBL5225255 0.88 KCNH2 (0.76) HDAC1KCNH2HDAC2HDAC3
SCHEMBL22738120 0.83 HDAC2 (0.71) HDAC1KCNH2HDAC2HDAC3
SCHEMBL20181677 0.81 HDAC2 (0.69) HDAC1KCNH2HDAC2HDAC3
SCHEMBL12193402 0.80 HDAC1 (0.59) HDAC1HDAC2HDAC3
SCHEMBL1639152 0.79 HDAC1 (0.68) HDAC1KCNH2HDAC2HDAC3
SCHEMBL1640302 0.79 HDAC1 (0.89) HDAC1KCNH2HDAC2HDAC3
SCHEMBL5224627 0.79 HDAC1 (0.56) HDAC1HDAC2HDAC3
SCHEMBL8161162 0.79 HDAC1 (0.70) HDAC1KCNH2HDAC2HDAC3
SCHEMBL1640845 0.79 HDAC1 (0.67) HDAC1KCNH2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501508-A1 INHIBITORS OF HISTONE DEACETYLASE Astrazeneca AB (SE) 2005-02-02 EP disclosed
WO-2003092686-A1 INHIBITORS OF HISTONE DEACETYLASE ASTRAZENECA AB (SE) 2003-11-13 WO disclosed