SCHEMBL6205635

SCHEMBL6205635

CC(=O)c1ccccc1CNc1ncnc2[nH]nnc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RPS6KB1 P23443 15/20 0.47
AURKA O14965 14/20 0.47
AURKB Q96GD4 3/20 0.45
CCNB2 O95067 3/20 0.42
CDK1 P06493 3/20 0.42
CCNB1 P14635 3/20 0.42
CCNB3 Q8WWL7 3/20 0.42
PDPK1 O15530 1/20 0.41
POLB P06746 1/20 0.38
DAPK3 O43293 1/20 0.37
JAK2 O60674 1/20 0.37
PRKD3 O94806 1/20 0.37
MAP4K4 O95819 1/20 0.37
PAK4 O96013 1/20 0.37
ABL1 P00519 1/20 0.37
CSF1R P07333 1/20 0.37
RET P07949 1/20 0.37
MET P08581 1/20 0.37
PDGFRB P09619 1/20 0.37
PIM1 P11309 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6205640 0.82 TSHR (0.43) RPS6KB1AURKAAURKBCCNB2CDK1
SCHEMBL4913008 0.82 AURKA (0.47) RPS6KB1AURKAAURKBCCNB2CDK1
SCHEMBL3445112 0.80 CDK2 (0.43) RPS6KB1AURKAAURKBCCNB2CDK1
SCHEMBL6205357 0.80 EGFR (0.54) RPS6KB1AURKAAURKBCCNB2CDK1
SCHEMBL3444022 0.79 CDK2 (0.50) RPS6KB1AURKAAURKBCCNB2CDK1
SCHEMBL3446179 0.77 CDK2 (0.48) CCNB2CDK1CCNB1CCNB3CDK7
SCHEMBL3444866 0.76 CDK1 (0.48) AURKACCNB2CDK1CCNB1CCNB3
SCHEMBL3444383 0.76 CDK2 (0.51) AURKACCNB2CDK1CCNB1CCNB3
SCHEMBL3444807 0.76 CDK2 (0.49) AURKBCDK1CCNB1PIM1GSK3B
SCHEMBL4913014 0.74 LMNA (0.65) KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539760-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2005-06-15 EP claimed
WO-2004018473-A2 AZAPURINE DERIVATIVES INSTITUTE OF EXPERIMENTAL BOTANY ASCR (CZ) 2004-03-04 WO claimed