SCHEMBL6207259

SCHEMBL6207259

O=C(/C=C\C(=O)Oc1ccc2cccccc1-2)Oc1ccc2cccccc1-2

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.53
HPGD P15428 2/20 0.53
MAPT P10636 1/20 0.53
HSD17B10 Q99714 1/20 0.53
FABP3 P05413 3/20 0.46
FABP5 Q01469 2/20 0.46
FABP7 O15540 1/20 0.46
TDP1 Q9NUW8 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
RXRA P19793 1/20 0.41
RXRB P28702 1/20 0.41
RXRG P48443 1/20 0.41
ALDH1A1 P00352 2/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
CYP2C9 P11712 1/20 0.40
BCAT2 O15382 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
GPR52 Q9Y2T5 1/20 0.40
HTT P42858 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5507667 0.83 ESR1 (0.58) KDM4EHPGDMAPTHSD17B10FABP3
SCHEMBL5169415 0.83 ESR1 (0.58) KDM4EHPGDMAPTHSD17B10FABP3
SCHEMBL29733244 0.80 FABP3 (0.49) KDM4EHPGDMAPTHSD17B10FABP3
SCHEMBL4389213 0.80 FABP3 (0.49) KDM4EHPGDMAPTHSD17B10FABP3
SCHEMBL35121 0.80 FABP3 (0.49) KDM4EHPGDMAPTHSD17B10FABP3
SCHEMBL27559161 0.79 BACE1 (0.58) KDM4EHPGDHSD17B10FABP3FABP5
Biphenyl SCHEMBL27827806 0.79 FABP3 (0.48) KDM4EHPGDMAPTHSD17B10FABP3
SCHEMBL4102451 0.78 KDM4E (0.43) KDM4EHPGDMAPTHSD17B10FABP3
SCHEMBL236823 0.77 FABP3 (0.53) KDM4EFABP3FABP5FABP7TDP1
SCHEMBL236822 0.77 FABP3 (0.53) KDM4EHPGDHSD17B10FABP3FABP5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546134-A1 PIPERAZINE SUBSTITUTED ARYL BENZODIAZEPINES ELI LILLY AND COMPANY (US) 2005-06-29 EP disclosed
WO-2004014895-A1 PIPERAZINE SUBSTITUTED ARYL BENZODIAZEPINES ELI LILLY AND COMPANY (US) 2004-02-19 WO disclosed