SCHEMBL6208008

SCHEMBL6208008

CC(C)(C)OC(=O)N1CC(Oc2ccc3ccccc3c2)CC1C(=O)O

nearest known ligand 0.63

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 14/20 0.47
UCHL1 P09936 1/20 0.44
P2RX3 P56373 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2437881 1.00 MCL1 (0.47) MCL1UCHL1P2RX3
SCHEMBL2434896 0.89 P2RX3 (0.50) MCL1UCHL1P2RX3
SCHEMBL192535 0.88 MCL1 (0.51) MCL1UCHL1P2RX3
SCHEMBL29015574 0.88 MCL1 (0.51) MCL1UCHL1P2RX3
SCHEMBL252870 0.88 MCL1 (0.51) MCL1UCHL1P2RX3
SCHEMBL23452261 0.88 MCL1 (0.51) MCL1UCHL1P2RX3
SCHEMBL6842708 0.88 MCL1 (0.51) MCL1UCHL1P2RX3
SCHEMBL192536 0.88 MCL1 (0.51) MCL1UCHL1P2RX3
SCHEMBL9544995 0.88 MCL1 (0.51) MCL1UCHL1P2RX3
SCHEMBL3188935 0.88 IKBKB (0.44) MCL1UCHL1P2RX3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1189612-A4 VLA-4 INHIBITOR COMPOUNDS DAIICHI SEIYAKU CO (JP) 2005-02-16 EP disclosed
EP-1189612-A1 VLA-4 INHIBITOR COMPOUNDS Daiichi Pharmaceutical Co., Ltd. (JP) 2002-03-27 EP disclosed
WO-2001000206-A1 VLA-4 INHIBITOR COMPOUNDS DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2001-01-04 WO disclosed