SCHEMBL6208539

SCHEMBL6208539

CCC(=O)Nc1nc(C)c(-c2ccnc(Nc3ccc(F)cc3)n2)s1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 9/20 0.64
CDK4 P11802 7/20 0.58
PLK1 P53350 3/20 0.58
CCNA2 P20248 1/20 0.58
AURKA O14965 5/20 0.58
CDK9 P50750 5/20 0.58
AURKB Q96GD4 5/20 0.58
CDK7 P50613 4/20 0.58
CDK1 P06493 3/20 0.58
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
WEE1 P30291 3/20 0.54
ALK Q9UM73 3/20 0.54
FLT3 P36888 2/20 0.54
CHEK1 O14757 1/20 0.54
DAPK3 O43293 1/20 0.54
JAK2 O60674 1/20 0.54
PRKD3 O94806 1/20 0.54
MAP4K4 O95819 1/20 0.54
PAK4 O96013 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1804658 0.92 CDK2 (0.64) CDK2CDK4PLK1CCNA2AURKA
SCHEMBL2073788 0.90 CDK2 (0.62) CDK2CDK4PLK1CCNA2AURKA
SCHEMBL6156585 0.84 CDK2 (0.71) CDK2CDK4PLK1CCNA2AURKA
SCHEMBL6209767 0.83 CDK2 (0.76) CDK2CDK4CCNA2AURKACDK9
SCHEMBL2285645 0.82 CDK2 (0.78) CDK2CDK4PLK1CCNA2AURKA
SCHEMBL2075966 0.82 CDK2 (0.65) CDK2CDK4PLK1CCNA2AURKA
SCHEMBL2074524 0.82 CDK2 (0.57) CDK2CDK4PLK1CCNA2AURKA
SCHEMBL4797854 0.81 CDK2 (0.67) CDK2CDK4PLK1CCNA2AURKA
SCHEMBL2073696 0.81 CDK2 (0.61) CDK2CDK4PLK1CCNA2AURKA
SCHEMBL4803422 0.80 CDK2 (0.65) CDK2CDK4PLK1CCNA2AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567522-A1 PYRIMIDINE COMPOUNDS Cyclacel Limited (GB) 2005-08-31 EP disclosed
WO-2004043953-A1 PYRIMIDINE COMPOUNDS CYCLACEL LIMITED (GB) 2004-05-27 WO disclosed