SCHEMBL6208965

SCHEMBL6208965

[CH2]C(=O)NCc1ccc(-c2cc(C(F)(F)F)nn2-c2ccc(OC)cc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 13/20 0.68
PTGS1 P23219 5/20 0.68
CYP2C9 P11712 2/20 0.62
CYP1A2 P05177 1/20 0.62
CYP3A4 P08684 1/20 0.62
TSHR P16473 1/20 0.62
CYP2C19 P33261 1/20 0.62
THPO P40225 1/20 0.62
BLM P54132 1/20 0.62
PMP22 Q01453 1/20 0.62
HIF1A Q16665 1/20 0.62
NPSR1 Q6W5P4 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5151993 0.91 PTGS2 (0.70) PTGS2PTGS1CYP2C9CYP1A2CYP3A4
SCHEMBL5148567 0.90 PTGS2 (0.68) PTGS2PTGS1CYP2C9CYP1A2CYP3A4
SCHEMBL5148824 0.89 PTGS2 (0.67) PTGS2PTGS1CYP2C9CYP1A2CYP3A4
SCHEMBL5149149 0.87 PTGS2 (0.64) PTGS2PTGS1CYP2C9CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL5150839 0.87 PTGS2 (0.64) PTGS2PTGS1CYP2C9CYP1A2CYP3A4
SCHEMBL5148913 0.84 PTGS2 (0.60) PTGS2PTGS1CYP2C9CYP1A2CYP3A4
SCHEMBL14504548 0.83 PTGS2 (0.67) PTGS2PTGS1CYP2C9CYP1A2CYP3A4
SCHEMBL14504542 0.83 PTGS2 (0.67) PTGS2PTGS1CYP2C9CYP1A2CYP3A4
SCHEMBL5147848 0.83 PTGS2 (0.73) PTGS2PTGS1CYP2C9CYP1A2CYP3A4
SCHEMBL5148972 0.83 PTGS2 (0.73) PTGS2PTGS1CYP2C9CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567503-A1 PYRAZOLE DERIVATIVES USEFUL AS COX-I INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2005-08-31 EP disclosed
WO-2004050632-A1 PYRAZOLE DERIVATIVES USEFUL AS COX-I INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-06-17 WO disclosed