SCHEMBL6209075

SCHEMBL6209075

CC(C)C[C@@H](Sc1ccc(-c2ccc(CN(C3CCC3)C3CCC3)cc2)cc1)C(=O)NCC#N

nearest known ligand 0.57

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSK P43235 13/20 0.45
CTSS P25774 13/20 0.45
CTSL P07711 11/20 0.43
CTSB P07858 10/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4703588 1.00 CTSK (0.45) CTSKCTSSCTSLCTSB
SCHEMBL4700894 0.99 CTSK (0.44) CTSKCTSSCTSLCTSB
SCHEMBL4702083 0.83 HRH3 (0.47) CTSKCTSSCTSLCTSB
SCHEMBL6209270 0.83 HRH3 (0.47) CTSKCTSSCTSLCTSB
SCHEMBL4701062 0.83 CTSK (0.47) CTSKCTSSCTSLCTSB
SCHEMBL4699985 0.82 CTSK (0.52) CTSKCTSSCTSLCTSB
SCHEMBL6271092 0.82 CTSK (0.52) CTSKCTSSCTSLCTSB
SCHEMBL4699909 0.81 CTSK (0.53) CTSKCTSSCTSLCTSB
SCHEMBL6211886 0.79 CTSK (0.67) CTSKCTSSCTSLCTSB
SCHEMBL4701868 0.79 CTSK (0.67) CTSKCTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1372655-A4 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA INC (CA) 2005-10-12 EP claimed
EP-1372655-A2 CATHEPSIN CYSTEINE PROTEASE INHIBITORS Merck Frosst Canada & Co. (CA) 2004-01-02 EP claimed
WO-2002069901-A2 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA & CO. (CA) 2002-09-12 WO claimed