SCHEMBL6209619

SCHEMBL6209619

Fc1cc(F)cc(-c2nc(-c3ccc(F)cc3F)n(Cc3ccccc3)c2Br)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.42
USP2 O75604 3/20 0.42
CYP1A2 P05177 3/20 0.42
CYP3A4 P08684 3/20 0.42
CYP2C9 P11712 3/20 0.42
MAPK1 P28482 3/20 0.42
CYP2C19 P33261 3/20 0.42
LMNA P02545 2/20 0.42
HSD17B10 Q99714 2/20 0.42
CYP11B2 P19099 1/20 0.39
GRM2 Q14416 1/20 0.38
KDM4E B2RXH2 2/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 3/20 0.38
HTT P42858 2/20 0.38
HK1 P19367 1/20 0.38
HKDC1 Q2TB90 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4830285 0.84 MAPT (0.41) ALDH1A1LMNAHSD17B10CYP11B2GRM2
SCHEMBL4833510 0.84 ALDH1A1 (0.43) ALDH1A1USP2CYP1A2CYP3A4CYP2C9
SCHEMBL6209919 0.80 MAPT (0.47) ALDH1A1MAPK1LMNAHSD17B10CYP11B2
SCHEMBL989287 0.72 TNF (0.45) ALDH1A1MAPK1LMNAHSD17B10CYP11B2
SCHEMBL27007784 0.68 KMT2A (0.44) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL990110 0.67 CYP2C19 (0.42) ALDH1A1CYP3A4CYP2C9CYP2C19CYP11B2
SCHEMBL4533975 0.66 ALDH1A1 (0.39) ALDH1A1USP2CYP1A2CYP3A4CYP2C9
SCHEMBL27007736 0.66 ALDH1A1 (0.48) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL5582032 0.64 TP53 (0.56) ALDH1A1CYP1A2CYP3A4CYP2C9MAPK1
SCHEMBL3522590 0.63 MAPK14 (0.56)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1554272-A1 BENZIMIDAZOLES AND BENZOTHIAZOLES AS INHIBITORS OF MAP KINASE ELI LILLY AND COMPANY (US) 2005-07-20 EP disclosed
WO-2004014900-A1 BENZIMIDAZOLES AND BENZOTHIAZOLES AS INHIBITORS OF MAP KINASE ELI LILLY AND COMPANY (US) 2004-02-19 WO disclosed