SCHEMBL6209689

SCHEMBL6209689

CCc1ccc(-c2c[nH]c(CCCN)c2NC(=O)OC(C)(C)C)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.38
PPARG P37231 2/20 0.33
ATR Q13535 1/20 0.33
PPARA Q07869 1/20 0.33
GLS O94925 1/20 0.33
FAAH O00519 1/20 0.33
JAK1 P23458 1/20 0.32
GRM2 Q14416 1/20 0.32
SREBF2 Q12772 1/20 0.32
SCN9A Q15858 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
HDAC3 O15379 2/20 0.32
HDAC8 Q9BY41 2/20 0.32
BRD4 O60885 1/20 0.32
CREBBP Q92793 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2909530 0.72 CNR2 (0.40) CYP17A1FAAHGRM2HDAC3HDAC8
SCHEMBL5868917 0.68 AAK1 (0.51) CYP17A1FAAHHDAC1
SCHEMBL10361607 0.68 CYP17A1 (0.61) CYP17A1PPARGPPARAFAAHHDAC3
SCHEMBL23092995 0.65 SMN1; SMN2 (0.43) CYP17A1PPARGCA1MEN1KMT2A
SCHEMBL30048842 0.65 CA2 (0.59) CA1CA2NAMPT
SCHEMBL18226965 0.65 CA1 (0.51) CA1CA2HDAC1NAMPTL3MBTL1
SCHEMBL5106837 0.65 CYP17A1 (0.57) CYP17A1PPARGPPARAGLSHDAC3
SCHEMBL21219242 0.64 AURKA (0.48) CYP17A1GLSCA1CA2HDAC3
SCHEMBL12740173 0.64 CYP17A1 (0.60) CYP17A1FAAHHDAC3HDAC8HDAC1
SCHEMBL25943313 0.64 CA1 (0.52) CA1CA2MEN1KMT2ANAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537099-A1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2005-06-08 EP disclosed
WO-2004018455-A1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2004-03-04 WO disclosed