SCHEMBL6210372

SCHEMBL6210372

CC(C)CC(NC(=O)c1ccc(C(F)(F)F)cc1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)C1=NC=CCC1=O

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CTSK P43235 16/20 0.52
CTSS P25774 2/20 0.41
CACNA1B Q00975 2/20 0.34
CCR1 P32246 1/20 0.34
CTSL P07711 1/20 0.33
KDM1A O60341 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6212234 0.92 CTSK (0.51) CTSKCTSSCCR1CTSL
SCHEMBL6213283 0.90 CTSK (0.61) CTSKCTSSCACNA1BCCR1CTSL
SCHEMBL6214785 0.89 CTSK (0.48) CTSKCTSSCTSL
SCHEMBL6213828 0.88 CTSK (0.57) CTSKCTSSCTSL
SCHEMBL6211235 0.88 CTSK (0.52) CTSKCTSSCCR1CTSL
SCHEMBL6210043 0.85 CTSK (0.51) CTSKCTSSCTSL
SCHEMBL6210782 0.84 CTSK (0.42) CTSKCTSSCCR1CTSL
SCHEMBL6210323 0.83 CTSK (0.49) CTSKCTSS
SCHEMBL6210601 0.83 CTSK (0.49) CTSKCTSSCTSL
SCHEMBL4037568 0.82 CTSK (0.58) CTSKCTSSCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP disclosed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO disclosed