SCHEMBL6219586

SCHEMBL6219586

NC(=O)OCCCCNc1c(N)cnc2cc(Br)ccc12

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.40
RXFP1 Q9HBX9 4/20 0.37
CSF1R P07333 1/20 0.36
BCHE P06276 6/20 0.36
ACHE P22303 6/20 0.36
GAA P10253 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
AURKB Q96GD4 1/20 0.33
EGFR P00533 1/20 0.33
ERBB2 P04626 1/20 0.33
SYK P43405 1/20 0.32
KDM4E B2RXH2 1/20 0.32
TOP2A P11388 1/20 0.32
RAB9A P51151 1/20 0.32
ENPP1 P22413 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL202429 0.87 MAPK1 (0.42) MAPK1RXFP1CSF1RBCHEACHE
SCHEMBL28888309 0.84 MEN1 (0.46) NPSR1TOP2A
SCHEMBL3867644 0.83 RXFP1 (0.40) MAPK1RXFP1CSF1RBCHEACHE
SCHEMBL19475071 0.81 TOP2A (0.41) MAPK1RXFP1GAANPSR1CYP1A2
SCHEMBL3169059 0.81 POLB (0.43) MAPK1RXFP1CSF1RCYP1A2CYP3A4
SCHEMBL3861875 0.81 CYP1A2 (0.42) MAPK1RXFP1CSF1RBCHEACHE
SCHEMBL4066480 0.81 NPC1 (0.41) BCHEACHEEGFRERBB2KDM4E
SCHEMBL5319030 0.81 MAPK1 (0.40) MAPK1RXFP1CSF1RBCHEACHE
SCHEMBL3861888 0.78 MAPK1 (0.41) MAPK1RXFP1CSF1RBCHEACHE
SCHEMBL4524933 0.78 ALDH1A1 (0.40) MAPK1RXFP1GAANPSR1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1590348-A1 ARYL / HETARYL SUBSTITUTED IMIDAZOQUINOLINES 3M Innovative Properties Company (US) 2005-11-02 EP disclosed
WO-2004058759-A1 ARYL / HETARYL SUBSTITUTED IMIDAZOQUINOLINES 3M INNOVATIVE PROPERTIES COMPANY (US) 2004-07-15 WO disclosed