Hexestrol Diphosphate

Hexestrol Diphosphate

SCHEMBL62206

CCC(c1ccc(OP(=O)(O)O)cc1)C(CC)c1ccc(OP(=O)(O)O)cc1

nearest known ligand 0.61

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BLM P54132 1/20 0.61
ESR1 P03372 2/20 0.54
HIF1A Q16665 1/20 0.54
CYP2C19 P33261 2/20 0.48
LMNA P02545 1/20 0.48
CYP1A2 P05177 1/20 0.48
PGR P06401 1/20 0.48
CHRM2 P08172 1/20 0.48
CYP3A4 P08684 1/20 0.48
ADORA3 P0DMS8 1/20 0.48
AR P10275 1/20 0.48
CYP2D6 P10635 1/20 0.48
MAPT P10636 1/20 0.48
CHRM1 P11229 1/20 0.48
CYP2C9 P11712 1/20 0.48
ALOX15 P16050 1/20 0.48
DRD1 P21728 1/20 0.48
TBXA2R P21731 1/20 0.48
PTGS1 P23219 1/20 0.48
SLC6A2 P23975 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hexestrol Diphosphate SCHEMBL4254504 1.00 BLM (0.61) BLMESR1HIF1ACYP2C19LMNA
SCHEMBL209725 0.93 ESR1 (0.61) BLMESR1HIF1ACYP2C19LMNA
SCHEMBL209724 0.93 ESR1 (0.61) BLMESR1HIF1ACYP2C19LMNA
Diethylstilbestrol Diphosphate SCHEMBL8153893 0.85 BLM (0.70) BLMESR1HIF1ACYP2C19LMNA
SCHEMBL12716935 0.84 BLM (0.54) BLMCYP2C19MAPTTDP1SRC
SCHEMBL4254509 0.81 ESR1 (0.54) BLMESR1HIF1ACYP2C19LMNA
SCHEMBL223266 0.79 SRC (0.54) BLMLMNASRCCA1CA2
SCHEMBL27342545 0.77 SRC (0.52) BLMLMNASRCCA1CA2
SCHEMBL329313 0.77 SRC (0.75) BLMCYP2C19CYP3A4SRCCA1
SCHEMBL924938 0.76 SRC (0.56) BLMCYP2C19SRCCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 7601 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260116861-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-04-30 US claimed
US-12522572-B2 Isoxazole hydroxamic acids as histone deacetylase 6 inhibitors THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-01-13 US claimed
WO-2025125890-A1 PROTEIN PHOSPHATASE 2A (PPA2) ANTAGONISTS FOR DENGUE TREATMENT CENTRO DE INVESTIGACIÓN Y DE ESTUDIOS AVANZADOS DEL I.P.N. (MX) 2025-06-19 WO claimed
US-20240343697-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2024-10-17 US claimed
US-20230228674-A1 Systems and Methods for Multianalyte Detection TRUVIAN SCIENCES, INC. 2023-07-20 US claimed
US-11345956-B2 Methods and compositions related to prostate cancer therapeutics THE JOHNS HOPKINS UNIVERSITY (US) 2022-05-31 US claimed
US-11207289-B2 Use of benzofuran lignans to induce IL-25 expression and suppress mammary tumor metastasis ACADEMIA SINICA (TW) 2021-12-28 US claimed
US-10953073-B2 XTEN conjugate compositions and methods of making same AMUNIX PHARMACEUTICALS, INC. (US) 2021-03-23 US claimed
US-20210060040-A1 CANNABINOID RECEPTOR MODULATORS ARENA PHARMACEUTICALS, INC. 2021-03-04 US claimed
EP-3191114-B1 OCCIDIOFUNGIN FORMULATIONS AND USES THEREOF UNIV MISSISSIPPI STATE (US) 2021-03-03 EP claimed
US-20060018933-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 US claimed
US-20060018934-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 US claimed
WO-2005067644-A2 CONJUGATED SMALL MOLECULES AMBIT BIOSCIENCES CORPORATION (US) 2005-07-28 WO claimed
US-20050153371-A1 Conjugated small molecules AMBIT BIOSCIENCES CORPORATION 2005-07-14 US claimed
US-20040092583-A1 Treatment for inhibiting neoplastic lesions SHANAHAN-PRENDERGAST ELIZABETH (IE) 2004-05-13 US claimed
EP-1351678-A2 TREATMENT FOR INHIBITING NEOPLASTIC LESIONS USING INCENSOLE AND/OR FURANOGERMACRENS Shanahan-Prendergast, Elizabeth (IE) 2003-10-15 EP claimed
WO-2002053138-A2 TREATMENT FOR INHIBITING NEOPLASTIC LESIONS USING INCENSOLE AND/OR FURANOGERMACRENS SHANAHAN-PRENDERGAST ELISABETH (IE) 2002-07-11 WO claimed
WO-1998044109-A1 CYTOSTATIN II HUMAN GENOME SCIENCES, INC. (US) 1998-10-08 WO claimed
EP-0759087-A1 COMPOSITIONS AND METHODS FOR TARGETING GENE DELIVERY VEHICLES CHIRON CORPORATION (US) 1997-02-26 EP claimed
WO-1995031566-A1 COMPOSITIONS AND METHODS FOR TARGETING GENE DELIVERY VEHICLES CHIRON VIAGENE, INC. (US) 1995-11-23 WO claimed