SCHEMBL6220975

SCHEMBL6220975

CCc1ccc(S(=O)(=O)O)cc1-c1nc(-c2ccccc2)oc1C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.42
LMNA P02545 1/20 0.42
TARBP2 Q15633 2/20 0.41
SLC9A1 P19634 1/20 0.41
PTPN2 P17706 2/20 0.39
PTPN1 P18031 2/20 0.39
PTPN5 P54829 2/20 0.39
RCE1 Q9Y256 1/20 0.39
USP1 O94782 1/20 0.39
USP19 O94966 1/20 0.39
WDR48 Q8TAF3 1/20 0.39
SMO Q99835 1/20 0.38
FAAH O00519 1/20 0.38
KCNH2 Q12809 1/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPK1 P28482 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
HPGD P15428 2/20 0.38
TSHR P16473 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5218987 0.75 TARBP2 (0.42) KDM4ELMNATARBP2PTPN2PTPN1
SCHEMBL6987242 0.75 NPC1 (0.39) KDM4ESLC9A1ALDH1A1NPSR1TSHR
SCHEMBL5736248 0.74 KDM4E (0.41) KDM4ELMNATARBP2SLC9A1PTPN1
SCHEMBL6703700 0.73 TARBP2 (0.46) KDM4ELMNATARBP2PTPN1SMO
SCHEMBL6220972 0.70 KDM4E (0.54) KDM4ELMNAPPARGPPARA
SCHEMBL2520539 0.70 FFAR1 (0.64) KDM4EKDRTP53PPARGPPARA
SCHEMBL6705288 0.70 TARBP2 (0.39) KDM4ELMNATARBP2PTPN1ALDH1A1
SCHEMBL6219926 0.70 KDM4E (0.40) KDM4ELMNATARBP2SLC9A1RCE1
SCHEMBL2089931 0.69 KDM4E (0.56) KDM4ETARBP2PTPN1USP1USP19
SCHEMBL28975550 0.68 KDM4E (0.52) KDM4ELMNAALDH1A1MAPK1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1597257-A1 OXAZOLE-DERIVATIVES AS PPAR AGONISTS PFIZER INC. (US) 2005-11-23 EP disclosed
US-20040209929-A1 Fused heteroaryl carboxylic acids as PPAR agonists AGOURON PHARMACEUTICALS, INC. 2004-10-21 US disclosed
WO-2004074284-A1 OXAZOLE-DERIVATIVES AS PPAR AGONISTS PFIZER INC. (US) 2004-09-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040209929-A1 Fused heteroaryl carboxylic acids as PPAR agonists PPARG, PPARA, PPARD KDM4E 2860/4885LMNA 3569/4885TARBP2 2474/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.