SCHEMBL6224902

SCHEMBL6224902

[CH2]c1ccc(-c2ccccn2)cc1CO

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CBFB Q13951 3/20 0.44
DHODH Q02127 1/20 0.43
CYP1A2 P05177 2/20 0.41
CCR1 P32246 2/20 0.41
CCR5 P51681 2/20 0.41
CCR8 P51685 2/20 0.41
KDM4E B2RXH2 2/20 0.41
LMNA P02545 1/20 0.41
POLB P06746 1/20 0.41
METAP1 P53582 1/20 0.41
BLM P54132 1/20 0.41
HIF1A Q16665 1/20 0.41
DOHH Q9BU89 1/20 0.41
P4HTM Q9NXG6 1/20 0.41
PDK2 Q15119 1/20 0.40
PRMT5 O14744 2/20 0.40
WDR77 Q9BQA1 1/20 0.40
P2RX7 Q99572 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP19A1 P11511 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14595530 0.85 CBFB (0.51) CBFBDHODHCYP1A2CCR1CCR5
SCHEMBL4539127 0.81 P2RX7 (0.54) CBFBDHODHCYP1A2CCR1CCR5
SCHEMBL21753409 0.77 CBFB (0.44) CBFBDHODHCYP1A2CCR1CCR5
SCHEMBL21753230 0.77 KDM4E (0.47) CBFBDHODHCYP1A2CCR1CCR5
SCHEMBL21769973 0.77 CBFB (0.53) CBFBDHODHCYP1A2CCR1CCR5
SCHEMBL5803772 0.77 ERN1 (0.48) CBFBCYP1A2KDM4EPOLBCYP2D6
SCHEMBL19794413 0.77 PDK2 (0.47) CBFBDHODHCYP1A2CCR1CCR5
SCHEMBL27357757 0.75 DCLRE1A (0.43) CYP1A2KDM4ELMNA
SCHEMBL30462045 0.72 KDM4E (0.50) CBFBDHODHCYP1A2CCR1CCR5
SCHEMBL533591 0.72 KDM4E (0.50) CBFBDHODHCYP1A2CCR1CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534676-A1 PIPERIDINETRIOL DERIVATIVES AS INHIBITORS OF GLYCOSYLCERAMIDE SYNTHASE Oxford GlycoSciences (UK) Limited (GB) 2005-06-01 EP disclosed
WO-2004007453-A1 PIPERIDINETRIOL DERIVATIVES AS INHIBITORS OF GLYCOSYLCERAMIDE SYNTHASE OXFORD GLYCOSCIENCES (UK) LTD (GB) 2004-01-22 WO disclosed