SCHEMBL6225664

SCHEMBL6225664

Brc1ccc2nccc(N3CCCCCN3)c2c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 5/20 0.64
HTT P42858 2/20 0.44
ADRB2 P07550 2/20 0.39
SLC22A12 Q96S37 5/20 0.38
CHKA P35790 1/20 0.37
NMT1 P30419 1/20 0.35
CHEK1 O14757 1/20 0.35
PIM1 P11309 1/20 0.35
AKT1 P31749 1/20 0.35
FLT3 P36888 1/20 0.35
PIM3 Q86V86 1/20 0.35
PKM P14618 1/20 0.35
ALOX15 P16050 1/20 0.35
CASP1 P29466 1/20 0.35
HSD17B10 Q99714 1/20 0.35
MEN1 O00255 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
KMT2A Q03164 1/20 0.35
ATM Q13315 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6206052 0.81 NCF1 (0.66) NCF1SLC22A12HSD17B10MEN1GAA
SCHEMBL731691 0.80 NCF1 (0.74) NCF1HTTADRB2SLC22A12CHKA
SCHEMBL3849006 0.78 NCF1 (1.00) NCF1HTTADRB2PIM1PIM3
SCHEMBL22715673 0.76 NCF1 (0.76) NCF1HTTADRB2SLC22A12CHKA
SCHEMBL29472100 0.76 NCF1 (0.76) NCF1HTTADRB2SLC22A12CHKA
SCHEMBL3847734 0.72 NCF1 (0.70) NCF1HTTADRB2SLC22A12PKM
SCHEMBL1543989 0.70 NCF1 (0.70) NCF1HTTADRB2CHKAPKM
SCHEMBL31737749 0.68 NCF1 (0.50) NCF1ADRB2MAPT
SCHEMBL21190487 0.68 NCF1 (0.67) NCF1HTTADRB2SLC22A12CHKA
SCHEMBL30734145 0.68 NCF1 (0.67) NCF1HTTADRB2MEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537121-A1 ANTIDEPRESSANT ARYLPIPERAZINE DERIVATIVES OF HETEROCYCLE-FUSED BENZODIOXANS Wyeth (US) 2005-06-08 EP disclosed
WO-2004024731-A1 ANTIDEPRESSANT ARYLPIPERAZINE DERIVATIVES OF HETEROCYCLE-FUSED BENZODIOXANS WYETH (US) 2004-03-25 WO disclosed