SCHEMBL6231003

SCHEMBL6231003

Clc1ccc(Nc2cc(Nc3ccccc3)nc3c(Br)cccc23)cc1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.48
MAPT P10636 1/20 0.48
NPY5R Q15761 1/20 0.47
POLA1 P09884 1/20 0.41
SLC2A1 P11166 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
POLB P06746 1/20 0.39
TP53 P04637 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
S1PR2 O95136 1/20 0.39
S1PR4 O95977 1/20 0.39
S1PR3 Q99500 1/20 0.39
ADORA3 P0DMS8 6/20 0.38
FADS1 O60427 1/20 0.37
TMEM97 Q5BJF2 4/20 0.36
SIGMAR1 Q99720 3/20 0.36
DRD3 P35462 2/20 0.36
CYP1A2 P05177 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6238034 0.89 GAA (0.45) GAAMAPTNPY5RPOLA1SLC2A1
SCHEMBL6235371 0.86 MAPT (0.42) GAAMAPTNPY5RPOLA1SLC2A1
SCHEMBL6233025 0.86 MAPT (0.42) GAAMAPTNPY5RPOLA1SLC2A1
SCHEMBL6235222 0.86 GAA (0.47) GAAMAPTNPY5RPOLA1SLC2A1
SCHEMBL6231640 0.86 SLC2A1 (0.48) GAAMAPTNPY5RSLC2A1MEN1
SCHEMBL6235120 0.86 NPY5R (0.47) MAPTNPY5RPOLA1SLC2A1MEN1
SCHEMBL6232210 0.84 MAPT (0.45) GAAMAPTMEN1KMT2APOLB
SCHEMBL6086853 0.84 GAA (0.50) GAAMAPTNPY5RPOLA1SLC2A1
SCHEMBL6238037 0.82 NPY5R (0.60) MAPTNPY5RPOLA1SLC2A1MEN1
SCHEMBL6089980 0.81 GAA (0.54) GAAMAPTNPY5RPOLA1SLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1430030-B1 N-TYPE CALCIUM CHANNEL ANTAGONISTS FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2005-05-18 EP disclosed