SCHEMBL6235064

SCHEMBL6235064

COc1cc([AsH2])ccc1C#N

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AR P10275 13/20 0.54
ALDH1A1 P00352 2/20 0.53
KDM4E B2RXH2 1/20 0.53
USP2 O75604 1/20 0.53
PGR P06401 1/20 0.50
IMPDH2 P12268 2/20 0.48
IMPDH1 P20839 1/20 0.48
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
HTR2A P28223 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2761994 0.82 ALDH1A1 (0.59) ARALDH1A1KDM4EUSP2PGR
SCHEMBL24476682 0.79 AR (0.54) ARALDH1A1KDM4EUSP2PGR
SCHEMBL1608900 0.79 AR (0.69) ARALDH1A1KDM4EUSP2PGR
SCHEMBL2614475 0.79 AR (0.69) ARALDH1A1KDM4EUSP2PGR
SCHEMBL1343373 0.78 ALDH1A1 (0.55) ARALDH1A1KDM4EUSP2PGR
SCHEMBL286644 0.78 AR (0.53) ARALDH1A1KDM4EUSP2PGR
SCHEMBL13560245 0.78 AR (0.53) ARALDH1A1KDM4EUSP2PGR
SCHEMBL551293 0.78 AR (0.53) ARALDH1A1KDM4EUSP2PGR
SCHEMBL7668281 0.78 AR (0.53) ARALDH1A1KDM4EUSP2PGR
SCHEMBL1642615 0.78 KDM4E (0.79) ARALDH1A1KDM4EUSP2PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1606268-A1 HETEROCYCLIC KINASE INHIBITORS Abbott Laboratories (US) 2005-12-21 EP disclosed
WO-2004076424-A1 HETEROCYCLIC KINASE INHIBITORS ABBOTT LABORATORIES (US) 2004-09-10 WO disclosed