SCHEMBL6235468

SCHEMBL6235468

C=CCOC(=O)N1C(=O)CC2NCC=C21

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.33
NPSR1 Q6W5P4 1/20 0.32
FAAH O00519 3/20 0.31
CYP3A4 P08684 1/20 0.31
TP53 P04637 1/20 0.31
TSHR P16473 1/20 0.31
GAA P10253 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
LMNA P02545 1/20 0.30
MAPK1 P28482 1/20 0.30
RAB9A P51151 1/20 0.30
MGLL Q99685 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4037917 0.73 TSHR (0.38) CYP19A1NPSR1FAAHCYP3A4TP53
SCHEMBL4041592 0.69 FAAH (0.35) CYP19A1FAAHCYP3A4TP53TSHR
SCHEMBL18485419 0.69 CYP3A4 (0.39) NPSR1FAAHCYP3A4TSHRLMNA
SCHEMBL4043279 0.67 FAAH (0.36) CYP19A1FAAHTP53TSHRGAA
SCHEMBL23812541 0.66 NPSR1 (0.40) CYP19A1NPSR1FAAHCYP3A4TSHR
SCHEMBL8521913 0.66 CYP3A4 (0.43) NPSR1CYP3A4TSHRMEN1KMT2A
SCHEMBL6930133 0.65 TSHR (0.37) NPSR1FAAHCYP3A4TSHRLMNA
SCHEMBL18485435 0.65 TSHR (0.37) NPSR1FAAHCYP3A4TSHRLMNA
SCHEMBL6235471 0.65 CYP19A1 (0.31) CYP19A1FAAH
SCHEMBL18485441 0.63 HTT (0.40) NPSR1FAAHCYP3A4TP53TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP disclosed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO disclosed