SCHEMBL623722

SCHEMBL623722

CN(C)C(=O)CN1CCC2(CC1)CC(Nc1nn3cc(-c4cccc(OC(F)(F)F)c4)nc3s1)C2

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 8/20 0.43
PIM3 Q86V86 2/20 0.37
MAPT P10636 1/20 0.36
F2RL3 Q96RI0 2/20 0.36
IRAK4 Q9NWZ3 1/20 0.36
JAK2 O60674 1/20 0.36
JAK3 P52333 1/20 0.36
PTK2 Q05397 1/20 0.36
KCNH2 Q12809 1/20 0.36
FYN P06241 1/20 0.36
PIM2 Q9P1W9 2/20 0.35
FLT3 P36888 1/20 0.35
TYRO3 Q06418 1/20 0.35
THRB P10828 1/20 0.35
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35
TRPA1 O75762 1/20 0.35
DGAT2 Q96PD7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625490 0.87 PIM1 (0.39) PIM1PIM3F2RL3KCNH2PIM2
SCHEMBL625296 0.85 F2RL3 (0.38) PIM1PIM3MAPTF2RL3IRAK4
SCHEMBL623721 0.85 FYN (0.48) PIM1PIM3KCNH2FYNPIM2
SCHEMBL625496 0.85 PIM1 (0.39) PIM1PIM3MAPTF2RL3IRAK4
SCHEMBL625561 0.83 PIM1 (0.49) PIM1PIM3F2RL3KCNH2PIM2
SCHEMBL623435 0.78 PIM1 (0.46) PIM1PIM3F2RL3KCNH2PIM2
SCHEMBL1944061 0.78 PIM1 (0.54) PIM1PIM3F2RL3KCNH2FYN
SCHEMBL1945312 0.77 FYN (0.45) PIM1MAPTF2RL3KCNH2FYN
SCHEMBL623873 0.76 IDH1 (0.44) PIM1MAPTKCNH2THRB
SCHEMBL624454 0.76 PIM1 (0.45) PIM1PIM3F2RL3KCNH2PIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed