SCHEMBL6237283

SCHEMBL6237283

Cc1cc2c(cc1C(NCc1cccc(F)c1)c1ccc(C(=O)O)cc1)C(C)(C)CCC2(C)C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 18/20 1.00
HNF4A P41235 4/20 1.00
RXRB P28702 5/20 0.45
RXRG P48443 4/20 0.45
RARG P13631 3/20 0.45
RARA P10276 2/20 0.45
RARB P10826 2/20 0.45
NR4A2 P43354 2/20 0.43
MEN1 O00255 1/20 0.43
CYP26A1 O43174 1/20 0.43
ABCB11 O95342 1/20 0.43
ESR1 P03372 1/20 0.43
PGR P06401 1/20 0.43
HTR1A P08908 1/20 0.43
ADRA2A P08913 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
CHRM1 P11229 1/20 0.43
DRD1 P21728 1/20 0.43
TBXA2R P21731 1/20 0.43
SLC6A2 P23975 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6242939 0.91 RXRA (0.83) RXRAHNF4ARXRBRXRGRARG
SCHEMBL6244445 0.90 RXRA (0.82) RXRAHNF4ARXRBRXRGRARG
SCHEMBL6239091 0.90 RXRA (0.81) RXRAHNF4ARXRBRXRGRARG
SCHEMBL6241831 0.78 RXRA (0.64) RXRAHNF4ARXRBRXRGRARG
SCHEMBL6239262 0.77 RXRA (0.64) RXRAHNF4ARXRBRXRGRARG
SCHEMBL6905874 0.74 RXRA (0.74) RXRAHNF4ARXRBRXRGRARG
SCHEMBL2685029 0.73 RXRA (0.76) RXRAHNF4ARXRBRXRGRARG
SCHEMBL6889522 0.73 RXRA (1.00) RXRAHNF4ARXRBRXRGRARG
SCHEMBL6242052 0.73 RXRA (0.77) RXRAHNF4ARXRBRXRGRARG
SCHEMBL6242056 0.73 RXRA (0.77) RXRAHNF4ARXRBRXRGRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005017185-A2 HEPATOCYTE NUCLEAR FACTOR 4α MODULATOR COMPOUNDS LIGAND PHARMCEUTICALS INCORPORATED (US) 2005-02-24 WO claimed
WO-2005017185-A2 HEPATOCYTE NUCLEAR FACTOR 4α MODULATOR COMPOUNDS LIGAND PHARMCEUTICALS INCORPORATED (US) 2005-02-24 WO disclosed