SCHEMBL623731

SCHEMBL623731

O=CCc1sc(-c2ccncc2)nc1Cc1ccc(Cl)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.47
MEN1 O00255 2/20 0.47
MAPT P10636 3/20 0.42
ALOX5 P09917 1/20 0.41
KDM4E B2RXH2 3/20 0.40
LMNA P02545 2/20 0.40
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
POLB P06746 1/20 0.39
LSS P48449 1/20 0.38
PTGDR2 Q9Y5Y4 3/20 0.37
ROCK2 O75116 3/20 0.37
ALDH1A1 P00352 2/20 0.37
GRK2 P25098 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
HPGD P15428 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL624460 0.82 MAPT (0.44) KMT2AMEN1MAPTALOX5KDM4E
SCHEMBL10288198 0.76 MEN1 (0.46) KMT2AMEN1MAPTALOX5KDM4E
SCHEMBL623525 0.76 KMT2A (0.49) KMT2AMEN1MAPTALOX5KDM4E
SCHEMBL5747523 0.76 RAB9A (0.52) KMT2AMEN1MAPTALOX5KDM4E
SCHEMBL624223 0.75 SMN1; SMN2 (0.58) KMT2AMEN1MAPTKDM4ELMNA
SCHEMBL622975 0.74 RAB9A (0.60) KMT2AMEN1MAPTKDM4ERAB9A
SCHEMBL623027 0.74 MAPT (0.47) KMT2AMEN1MAPTALOX5KDM4E
SCHEMBL623495 0.73 CDC7 (0.51) KMT2AMEN1MAPTALOX5KDM4E
Hydrochloric Acid SCHEMBL623549 0.73 MAPT (0.46) KMT2AMEN1MAPTALOX5KDM4E
SCHEMBL27905821 0.72 MAPT (0.54) KMT2AMEN1MAPTKDM4ERAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2603214-A1 HETEROARYLS AND USES THEREOF Millennium Pharmaceuticals, Inc. (US) 2013-06-19 EP disclosed
WO-2012021696-A1 HETEROARYLS AND USES THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2012-02-16 WO disclosed