SCHEMBL6239207

SCHEMBL6239207

CC(C)S(=O)(=O)NC1CCC=C1c1ccc(-c2cc(F)cc(F)c2)cc1

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GRIA4 P48058 3/20 0.44
GRIA2 P42262 14/20 0.40
KCNH2 Q12809 3/20 0.35
CYP2C19 P33261 1/20 0.35
CXCR2 P25025 1/20 0.35
NPY5R Q15761 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6240181 0.93 GRIA4 (0.45) GRIA4GRIA2KCNH2CYP2C19NPY5R
SCHEMBL6240609 0.92 GRIA4 (0.48) GRIA4GRIA2CYP2C19CXCR2NPY5R
SCHEMBL6243805 0.84 GRIA4 (0.44) GRIA4GRIA2KCNH2
SCHEMBL6240540 0.84 ADAM17 (0.41) GRIA4GRIA2
SCHEMBL6242243 0.82 CXCR2 (0.37) GRIA4GRIA2CXCR2
SCHEMBL6241425 0.82 GRIA4 (0.48) GRIA4GRIA2CXCR2
SCHEMBL6239214 0.81 CYP11B1 (0.40) CYP2C19NPY5R
SCHEMBL6242831 0.80 GRIA2 (0.52) GRIA4GRIA2KCNH2
SCHEMBL6245808 0.80 CA12 (0.41) GRIA2KCNH2
SCHEMBL6240728 0.78 GRIA4 (0.39) GRIA4GRIA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1395550-B1 CYCLOALKENYLSULFONAMIDE DERIVATIVES LILLY CO ELI (US) 2005-06-29 EP disclosed
US-20040157817-A1 Cycloalkenylsulfonamide derivatives CANTELL BUDDY EUGENE (US) 2004-08-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040157817-A1 Cycloalkenylsulfonamide derivatives GRIN2B, GRIN2A, GRIN1 GRIA4 14/4885GRIA2 7/4885KCNH2 552/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.