SCHEMBL6239333

SCHEMBL6239333

Nc1ccc2[nH]c(N3CCOCC3)nc2c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.64
SMN1; SMN2 Q16637 4/20 0.48
MAPT P10636 3/20 0.48
NPC1 O15118 3/20 0.48
RAB9A P51151 3/20 0.48
GAA P10253 2/20 0.48
KDM4E B2RXH2 1/20 0.47
BCHE P06276 1/20 0.44
ACHE P22303 1/20 0.44
PIK3CA P42336 3/20 0.43
HTR3A P46098 1/20 0.43
PIK3R1 P27986 1/20 0.42
MTOR P42345 1/20 0.42
POLB P06746 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
TRPC3 Q13507 1/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
NFKB1 P19838 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6232538 0.86 BCHE (0.59) TP53SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL6231870 0.85 BCHE (0.62) TP53SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL31154250 0.82 TP53 (0.44) TP53SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL6236251 0.82 NPC1 (0.58) TP53MAPTNPC1RAB9AGAA
SCHEMBL19145306 0.82 TP53 (0.64) TP53SMN1; SMN2NPC1RAB9AGAA
SCHEMBL1663221 0.80 PARP1 (0.52) TP53SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL19117309 0.79 TP53 (0.59) TP53SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL26226732 0.79 TP53 (0.59) TP53SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL2674838 0.78 TP53 (1.00) TP53SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL27938349 0.78 HTR2B (0.49) TP53MAPTBCHEACHEHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004092181-A9 HETEROCYCLIC MCHR1 ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2005-01-27 WO disclosed