Pazelliptine

Pazelliptine

SCHEMBL62441

CCN(CC)CCCNc1nccc2c(C)c3[nH]c4ccncc4c3cc12

nearest known ligand 0.73

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIT P10721 8/20 0.73
PDGFRA P16234 2/20 0.42
FGFR3 P22607 2/20 0.42
NQO1 P15559 1/20 0.41
GSK3A P49840 1/20 0.41
GSK3B P49841 1/20 0.41
NPSR1 Q6W5P4 3/20 0.41
ALDH1A1 P00352 2/20 0.41
PAX8 Q06710 1/20 0.41
GAA P10253 2/20 0.40
BRAF P15056 1/20 0.40
TP53 P04637 2/20 0.39
TERT O14746 1/20 0.39
NSD2 O96028 1/20 0.39
KDM4E B2RXH2 2/20 0.39
MEN1 O00255 2/20 0.39
NR3C1 P04150 2/20 0.39
POLB P06746 2/20 0.39
MAPT P10636 2/20 0.39
RECQL P46063 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pazelliptine SCHEMBL29376377 1.00 KIT (0.73) KITPDGFRAFGFR3NQO1GSK3A
Pazelliptine SCHEMBL1230910 0.99 KIT (0.72) KITPDGFRAFGFR3NQO1GSK3A
Pazelliptine SCHEMBL1230570 0.98 KIT (0.71) KITPDGFRAFGFR3NQO1GSK3A
SCHEMBL2311857 0.94 KIT (0.65) KITPDGFRAFGFR3NPSR1ALDH1A1
SCHEMBL13498771 0.93 KIT (0.66) KITPDGFRAFGFR3NQO1GSK3A
SCHEMBL12387163 0.91 KIT (0.61) KITPDGFRAFGFR3NPSR1ALDH1A1
SCHEMBL2308783 0.90 KIT (0.59) KITPDGFRAFGFR3NPSR1ALDH1A1
SCHEMBL2308791 0.86 KIT (0.55) KITPDGFRAFGFR3NPSR1ALDH1A1
SCHEMBL2311605 0.86 KIT (0.54) KITPDGFRAFGFR3NPSR1ALDH1A1
SCHEMBL1065037 0.85 KIT (0.78) KITPDGFRAFGFR3NQO1GSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 8614 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260116861-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-04-30 US claimed
US-12522572-B2 Isoxazole hydroxamic acids as histone deacetylase 6 inhibitors THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-01-13 US claimed
US-20240343697-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2024-10-17 US claimed
US-11345956-B2 Methods and compositions related to prostate cancer therapeutics THE JOHNS HOPKINS UNIVERSITY (US) 2022-05-31 US claimed
US-11207289-B2 Use of benzofuran lignans to induce IL-25 expression and suppress mammary tumor metastasis ACADEMIA SINICA (TW) 2021-12-28 US claimed
US-20210060040-A1 CANNABINOID RECEPTOR MODULATORS ARENA PHARMACEUTICALS, INC. 2021-03-04 US claimed
EP-3191114-B1 OCCIDIOFUNGIN FORMULATIONS AND USES THEREOF UNIV MISSISSIPPI STATE (US) 2021-03-03 EP claimed
US-20200289454-A1 USE OF BENZOFURAN LIGNANS TO INDUCE IL-25 EXPRESSION AND SUPPRESS MAMMARY TUMOR METASTASIS Yang, Ning-Sun (TW) 2020-09-17 US claimed
US-20200270362-A1 MSLN TARGETING TRISPECIFIC PROTEINS AND METHODS OF USE HARPOON THERAPEUTICS, INC. 2020-08-27 US claimed
US-10265374-B2 Occidiofungin formations and uses thereof MISSISSIPPI STATE UNIVERSITY (US) 2019-04-23 US claimed
US-20060018933-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 US claimed
WO-2005023255-A2 USE OF INDOLE-DERIVED COMPOUNDS FOR THE PREPARATION OF A MEDICAMENT THAT CAN BE USED TO TREAT DISEASES RELATED TO THE SPLICING PROCESS CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2005-03-17 WO claimed
US-20040092583-A1 Treatment for inhibiting neoplastic lesions SHANAHAN-PRENDERGAST ELIZABETH (IE) 2004-05-13 US claimed
EP-1351678-A2 TREATMENT FOR INHIBITING NEOPLASTIC LESIONS USING INCENSOLE AND/OR FURANOGERMACRENS Shanahan-Prendergast, Elizabeth (IE) 2003-10-15 EP claimed
WO-2002053138-A2 TREATMENT FOR INHIBITING NEOPLASTIC LESIONS USING INCENSOLE AND/OR FURANOGERMACRENS SHANAHAN-PRENDERGAST ELISABETH (IE) 2002-07-11 WO claimed
EP-1085891-A1 MULTIBINDING INHIBITORS OF TOPOISOMERASE Advanced Medicine, Inc. (US) 2001-03-28 EP claimed
WO-1999064054-A9 MULTIBINDING INHIBITORS OF TOPOISOMERASE ADVANCED MEDICINE INC (US) 2000-03-02 WO claimed
WO-1999064054-A1 MULTIBINDING INHIBITORS OF TOPOISOMERASE ADVANCED MEDICINE, INC. (US) 1999-12-16 WO claimed
EP-0393575-B1 Neoplasia treatment compositions containing antineoplastic agent and side-effect reducing protective agent SEARLE & CO (US) 1994-03-16 EP claimed
EP-0393575-A1 Neoplasia treatment compositions containing antineoplastic agent and side-effect reducing protective agent G.D. Searle & Co. (US) 1990-10-24 EP claimed