SCHEMBL6246331

SCHEMBL6246331

CC(C)CC(C(=O)NCC#N)c1cccc(-c2ccccc2F)c1

nearest known ligand 0.79

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSK P43235 20/20 0.79
CTSS P25774 14/20 0.79
CTSL P07711 12/20 0.79
CTSB P07858 7/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4715050 0.88 CTSK (1.00) CTSKCTSSCTSLCTSB
SCHEMBL4714956 0.88 CTSK (0.77) CTSKCTSSCTSLCTSB
SCHEMBL4712626 0.88 CTSK (0.77) CTSKCTSSCTSLCTSB
SCHEMBL6245127 0.88 CTSK (0.77) CTSKCTSSCTSLCTSB
SCHEMBL4712376 0.86 CTSK (0.82) CTSKCTSSCTSLCTSB
SCHEMBL4711738 0.86 CTSK (0.74) CTSKCTSSCTSLCTSB
SCHEMBL14290542 0.85 CTSK (0.84) CTSKCTSSCTSLCTSB
SCHEMBL4712315 0.82 CTSK (0.82) CTSKCTSSCTSLCTSB
SCHEMBL4716587 0.82 CTSK (0.82) CTSKCTSSCTSLCTSB
SCHEMBL4714892 0.82 CTSK (0.82) CTSKCTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1248612-A4 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS MERCK FROSST CANADA INC (CA) 2005-09-07 EP claimed
EP-1248612-A1 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS MERCK FROSST CANADA INC. (CA) 2002-10-16 EP claimed
WO-2001049288-A1 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS MERCK FROSST CANADA & CO. (CA) 2001-07-12 WO claimed
EP-1248612-A4 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS MERCK FROSST CANADA INC (CA) 2005-09-07 EP disclosed
EP-1248612-A1 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS MERCK FROSST CANADA INC. (CA) 2002-10-16 EP disclosed
WO-2001049288-A1 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS MERCK FROSST CANADA & CO. (CA) 2001-07-12 WO disclosed