SCHEMBL624880

SCHEMBL624880

FCCC(Nc1nn2c(-c3cccc(OC(F)(F)F)c3)cnc2s1)C1CCNCC1

nearest known ligand 0.51

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 19/20 0.51
KCNH2 Q12809 2/20 0.44
DYRK1A Q13627 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL624007 0.87 PIM1 (0.51) PIM1KCNH2DYRK1A
SCHEMBL624838 0.85 PIM1 (0.48) PIM1KCNH2DYRK1A
SCHEMBL625502 0.82 PIM1 (0.69) PIM1KCNH2
Hydrochloric Acid SCHEMBL625022 0.82 FYN (0.58) PIM1KCNH2
SCHEMBL623848 0.79 DYRK1A (0.47) PIM1KCNH2DYRK1A
SCHEMBL624032 0.78 PIM1 (0.47) PIM1KCNH2DYRK1A
SCHEMBL1945251 0.78 FYN (0.64) PIM1KCNH2
SCHEMBL1945309 0.76 FYN (0.71) PIM1KCNH2
SCHEMBL625516 0.76 PIM1 (0.57) PIM1KCNH2DYRK1A
SCHEMBL28944695 0.76 DYRK1A (0.54) PIM1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed