SCHEMBL624032

SCHEMBL624032

FC(F)(F)c1cccc(-c2cnc3sc(NC(CC4CC4)C4CCNCC4)nn23)c1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 9/20 0.47
FYN P06241 7/20 0.45
KCNH2 Q12809 2/20 0.41
DYRK1A Q13627 3/20 0.40
DYRK2 Q92630 3/20 0.40
CCNA2 P20248 2/20 0.40
CDK2 P24941 2/20 0.40
CDK5 Q00535 2/20 0.40
CDK5R1 Q15078 2/20 0.40
DYRK1B Q9Y463 2/20 0.40
CCNT1 O60563 1/20 0.40
CDK9 P50750 1/20 0.40
MKNK1 Q9BUB5 1/20 0.40
AURKA O14965 1/20 0.39
FLT3 P36888 1/20 0.39
GSK3B P49841 1/20 0.39
PIM3 Q86V86 1/20 0.39
PIM2 Q9P1W9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL623848 0.90 DYRK1A (0.47) PIM1FYNKCNH2DYRK1ADYRK2
SCHEMBL623881 0.82 FYN (0.60) PIM1FYNKCNH2MKNK1PIM3
SCHEMBL17004609 0.80 FYN (0.67) PIM1FYNKCNH2DYRK1ADYRK2
SCHEMBL624880 0.78 PIM1 (0.51) PIM1KCNH2DYRK1A
SCHEMBL1946065 0.74 FYN (0.68) PIM1FYNKCNH2MKNK1PIM2
SCHEMBL1945221 0.74 FYN (0.76) PIM1FYNKCNH2DYRK1ADYRK2
SCHEMBL27815771 0.74 DYRK1A (0.53) PIM1FYNKCNH2DYRK1ADYRK2
SCHEMBL624030 0.74 FYN (0.59) PIM1FYNKCNH2MKNK1PIM3
SCHEMBL625548 0.73 FYN (0.52) PIM1FYNKCNH2DYRK1ADYRK2
SCHEMBL623882 0.73 DYRK1A (0.46) PIM1FYNKCNH2DYRK1ADYRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed