SCHEMBL6250185

SCHEMBL6250185

CSc1cc2c(cn1)c(=O)[nH]n2C

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE9A O76083 2/20 0.35
KDM4E B2RXH2 2/20 0.35
TP53 P04637 1/20 0.35
ALDH1A1 P00352 1/20 0.33
GLA P06280 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19493638 0.77 KDM4E (0.37) KDM4ETP53ALDH1A1HPGDMAPT
SCHEMBL1813535 0.68 MEN1 (0.42) PDE9AKDM4ETP53ALDH1A1GLA
SCHEMBL11622505 0.67 KDM4E (0.32) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL24046743 0.67 ADORA2A (0.53)
SCHEMBL24835534 0.66 ALDH1A1 (0.43) PDE9AKDM4EALDH1A1GLAGAA
SCHEMBL6244757 0.66 ADORA2A (0.35)
SCHEMBL11623684 0.65 KDM4E (0.32) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL2267451 0.63 KDM4E (0.44) KDM4ETP53ALDH1A1GAAHPGD
SCHEMBL29530274 0.63 KDM4E (0.40) KDM4ETP53
SCHEMBL22056718 0.62 PARP1 (0.50) PDE9AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1432714-A4 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2005-10-19 EP disclosed
EP-1432714-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2004-06-30 EP disclosed
WO-2003029209-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2003-04-10 WO disclosed