SCHEMBL625243

SCHEMBL625243

CN(C)c1cccc(-c2cnc3sc(NC4CC5(CCN(C(=O)OC(C)(C)C)CC5)C4)nn23)c1

nearest known ligand 0.60

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
FYN P06241 16/20 0.60
JAK2 O60674 1/20 0.40
JAK3 P52333 1/20 0.40
PTK2 Q05397 1/20 0.40
CDK9 P50750 1/20 0.39
NAMPT P43490 1/20 0.38
SCD5 Q86SK9 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL624036 0.88 FYN (0.46) FYNCDK9
SCHEMBL623828 0.88 FYN (0.46) FYNCDK9
SCHEMBL625495 0.86 PIM1 (0.46) FYN
SCHEMBL625540 0.83 FYN (0.68) FYN
SCHEMBL624057 0.81 FYN (0.60) FYNJAK2JAK3PTK2
SCHEMBL625491 0.80 NAMPT (0.41) CDK9NAMPT
SCHEMBL625407 0.79 PIK3CA (0.45) FYNCDK9NAMPT
SCHEMBL624945 0.77 FYN (0.49) FYN
SCHEMBL624433 0.76 FYN (0.47) FYNJAK2JAK3PTK2
SCHEMBL623872 0.76 FYN (0.52) FYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed