SCHEMBL625292

SCHEMBL625292

FC(F)(F)Oc1cccc(-c2cn3nc(NC4CCOCC4)sc3n2)c1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 15/20 0.53
DYRK1A Q13627 1/20 0.47
PIM3 Q86V86 1/20 0.44
KCNH2 Q12809 1/20 0.43
F2RL3 Q96RI0 2/20 0.42
PIM2 Q9P1W9 4/20 0.42
CSNK1E P49674 1/20 0.42
FLT3 P36888 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1945312 0.91 FYN (0.45) PIM1KCNH2F2RL3PIM2FLT3
SCHEMBL1944061 0.90 PIM1 (0.54) PIM1PIM3KCNH2F2RL3PIM2
SCHEMBL626259 0.89 PIM1 (0.53) PIM1KCNH2F2RL3PIM2FLT3
SCHEMBL623435 0.88 PIM1 (0.46) PIM1PIM3KCNH2F2RL3PIM2
Hydrochloric Acid SCHEMBL625023 0.88 PIM1 (0.45) PIM1PIM3KCNH2F2RL3PIM2
SCHEMBL1944168 0.86 PIM1 (0.55) PIM1DYRK1APIM3KCNH2F2RL3
SCHEMBL625501 0.83 PIM1 (0.43) PIM1KCNH2F2RL3PIM2FLT3
SCHEMBL623873 0.82 IDH1 (0.44) PIM1DYRK1AKCNH2
SCHEMBL625561 0.81 PIM1 (0.49) PIM1PIM3KCNH2F2RL3PIM2
SCHEMBL1945253 0.81 PIM1 (0.47) PIM1PIM3KCNH2F2RL3PIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed