SCHEMBL6252966

SCHEMBL6252966

C=CC[C@]12CC[C@]3(C)[C@@H](F)[C@H](O)C[C@H]3[C@@H]1CCc1cc(O)ccc12.C=C[C@]12CC[C@]3(C)[C@@H](F)[C@H](O)C[C@H]3[C@@H]1CCc1cc(O)ccc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 12/20 0.45
ESR1 P03372 5/20 0.45
ESR2 Q92731 5/20 0.45
PGR P06401 3/20 0.45
AR P10275 2/20 0.36
LMNA P02545 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
HIF1A Q16665 1/20 0.36
SHBG P04278 1/20 0.36
SERPINA6 P08185 1/20 0.36
PTGS1 P23219 1/20 0.36
SLC6A4 P31645 1/20 0.36
SNCA P37840 1/20 0.36
SLC6A3 Q01959 1/20 0.36
OR51E2 Q9H255 1/20 0.36
UGT1A10 Q9HAW8 1/20 0.36
OPRM1 P35372 2/20 0.33
OPRD1 P41143 2/20 0.33
OPRK1 P41145 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4588410 0.94 NR3C1 (0.49) NR3C1ESR1ESR2PGRAR
SCHEMBL6027234 0.91 ESR1 (0.44) NR3C1ESR1ESR2PGRAR
SCHEMBL6028199 0.91 ESR1 (0.44) NR3C1ESR1ESR2PGRAR
SCHEMBL1829051 0.91 ESR1 (0.44) NR3C1ESR1ESR2PGRAR
SCHEMBL12513381 0.82 NR3C1 (0.50) NR3C1ESR1ESR2PGRAR
SCHEMBL4587569 0.81 ESR1 (0.44) NR3C1ESR1ESR2PGRAR
SCHEMBL4587563 0.81 ESR1 (0.44) NR3C1ESR1ESR2PGRAR
SCHEMBL4589474 0.75 NR3C1 (0.53) NR3C1ESR1ESR2PGRAR
SCHEMBL4588414 0.72 ESR1 (0.41) NR3C1ESR1ESR2PGRAR
SCHEMBL6232274 0.72 ESR1 (0.37) NR3C1ESR1ESR2PGRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1517914-B1 9-ALPHA-SUBSTITUTED ESTRATRIENES AS SELECTIVELY ACTIVE ESTROGEN SCHERING AG (DE) 2005-08-31 EP claimed