SCHEMBL625465

SCHEMBL625465

COc1cncc(-c2cn3nc(NC4CCNCC4)sc3n2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FYN P06241 5/20 0.52
BRD4 O60885 1/20 0.42
BRD2 P25440 1/20 0.42
BRD3 Q15059 1/20 0.42
BRDT Q58F21 1/20 0.42
ATAD2 Q6PL18 1/20 0.42
DYRK1A Q13627 1/20 0.40
SYK P43405 1/20 0.40
F2RL3 Q96RI0 2/20 0.39
BRAF P15056 1/20 0.39
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
CYP2C19 P33261 1/20 0.39
MKNK1 Q9BUB5 1/20 0.38
PIK3CG P48736 1/20 0.38
TYRO3 Q06418 1/20 0.38
CYP1A2 P05177 2/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1944169 0.90 FYN (0.53) FYNSYKF2RL3BRAFPDE4A
SCHEMBL2253571 0.88 FYN (0.52) FYNSYKF2RL3BRAFPDE4A
SCHEMBL624392 0.86 FYN (0.54) FYNSYKF2RL3MKNK1TYRO3
SCHEMBL624431 0.84 FYN (0.48) FYNDYRK1ASYKF2RL3BRAF
SCHEMBL625464 0.80 FYN (0.78) FYN
SCHEMBL1945185 0.80 FYN (0.58) FYNF2RL3MKNK1PIK3CGMAPT
SCHEMBL1947142 0.76 FYN (0.68) FYNF2RL3
SCHEMBL1945374 0.76 FYN (0.64) FYNF2RL3MKNK1PIK3CGTP53
Hydrochloric Acid SCHEMBL625023 0.76 PIM1 (0.45) F2RL3TYRO3
SCHEMBL625236 0.75 MAP3K12 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed