SCHEMBL625503

SCHEMBL625503

CN(c1nn2c(-c3cccc(OC(F)(F)F)c3)cnc2s1)C1CCNCC1

nearest known ligand 0.52

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 11/20 0.52
DYRK1A Q13627 8/20 0.48
KCNH2 Q12809 2/20 0.46
FYN P06241 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1945252 0.94 DYRK1A (0.52) PIM1DYRK1AKCNH2FYN
SCHEMBL624008 0.87 PIM1 (0.56) PIM1DYRK1AKCNH2
SCHEMBL623882 0.86 DYRK1A (0.46) PIM1DYRK1AKCNH2FYN
SCHEMBL623013 0.85 PIM1 (0.47) PIM1DYRK1AKCNH2FYN
SCHEMBL2251446 0.80 DYRK1A (0.49) PIM1DYRK1AKCNH2FYN
Hydrochloric Acid SCHEMBL625022 0.79 FYN (0.58) PIM1KCNH2FYN
SCHEMBL1945068 0.79 DYRK1A (0.55) PIM1DYRK1AFYN
SCHEMBL624007 0.78 PIM1 (0.51) PIM1DYRK1AKCNH2FYN
SCHEMBL1944553 0.78 DYRK1A (0.47) PIM1DYRK1AFYN
SCHEMBL625502 0.78 PIM1 (0.69) PIM1KCNH2FYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed