SCHEMBL625602

SCHEMBL625602

COc1cncc(-c2c(C)nc3sc(NC(C4CCNCC4)S(C)(=O)=O)nn23)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FYN P06241 8/20 0.39
BRD4 O60885 1/20 0.34
BRD2 P25440 1/20 0.34
BRD3 Q15059 1/20 0.34
BRDT Q58F21 1/20 0.34
ATAD2 Q6PL18 1/20 0.34
PI4KA P42356 1/20 0.33
TYRO3 Q06418 1/20 0.32
GSK3B P49841 1/20 0.32
DYRK1A Q13627 1/20 0.32
BRAF P15056 1/20 0.31
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31
PIK3CG P48736 1/20 0.31
MMP1 P03956 1/20 0.31
MMP2 P08253 1/20 0.31
MMP3 P08254 1/20 0.31
MMP7 P09237 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL625478 0.86 FYN (0.55) FYNPIK3CA
SCHEMBL626614 0.79 FYN (0.57) FYN
SCHEMBL626613 0.79 FYN (0.36) FYNBRD4BRD2BRD3BRDT
SCHEMBL625600 0.74 FYN (0.53) FYNPI4KAGSK3B
SCHEMBL624838 0.70 PIM1 (0.48) FYNDYRK1A
SCHEMBL626615 0.67 FYN (0.57) FYNBRD4BRD2BRD3BRDT
SCHEMBL624884 0.67 FYN (0.51) FYNDYRK1A
SCHEMBL625464 0.66 FYN (0.78) FYN
SCHEMBL624391 0.64 FYN (0.79) FYN
SCHEMBL624390 0.63 FYN (0.52) FYNPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed