SCHEMBL6259620

SCHEMBL6259620

CCn1c(=O)[nH]c(=O)c2cc(C(=O)O)ccc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.53
KMT2A Q03164 4/20 0.53
KDM4E B2RXH2 9/20 0.53
HPGD P15428 6/20 0.53
HSD17B10 Q99714 3/20 0.53
TSHR P16473 2/20 0.53
B3GNT2 Q9NY97 1/20 0.48
HDAC1 Q13547 2/20 0.47
HDAC8 Q9BY41 2/20 0.47
HDAC6 Q9UBN7 2/20 0.47
GAA P10253 2/20 0.47
HCAR3 P49019 1/20 0.46
MAPT P10636 3/20 0.44
MEN1 O00255 3/20 0.44
THRB P10828 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
HTT P42858 2/20 0.43
RXFP1 Q9HBX9 1/20 0.43
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6840351 0.82 ALDH1A1 (0.72) ALDH1A1KMT2AKDM4EHPGDHSD17B10
SCHEMBL8922345 0.81 HPGD (0.65) ALDH1A1KMT2AKDM4EHPGDHSD17B10
SCHEMBL29629313 0.81 HPGD (0.65) ALDH1A1KMT2AKDM4EHPGDHSD17B10
SCHEMBL29629312 0.81 HPGD (0.65) ALDH1A1KMT2AKDM4EHPGDHSD17B10
SCHEMBL6243935 0.81 KDM4E (0.56) ALDH1A1KMT2AKDM4EHPGDHSD17B10
Hydrochloric Acid SCHEMBL8920877 0.80 HPGD (0.63) ALDH1A1KMT2AKDM4EHPGDHSD17B10
SCHEMBL21839442 0.79 B3GNT2 (0.72) ALDH1A1KMT2AKDM4EHPGDHSD17B10
SCHEMBL17434512 0.77 KDM4E (0.55) ALDH1A1KMT2AKDM4EHPGDHSD17B10
SCHEMBL6393500 0.76 PARG (0.45) ALDH1A1KMT2AKDM4EHPGDHSD17B10
SCHEMBL9747639 0.76 PTGER4 (0.59) ALDH1A1KMT2AKDM4EHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1531904-A1 COMBINATION OF AN ALLOSTERIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH A SELECTIVE INHIBITOR OF CYCLOOXYGENASE-2 THAT IS NOT CELECOXIB OR VALDECOXIB Warner-Lambert Company LLC (US) 2005-05-25 EP disclosed
WO-2004007024-A1 COMBINATION OF AN ALLOSTERIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH A SELECTIVE INHIBITOR OF CYCLOOXYGENASE-2 THAT IS NOT CELECOXIB OR VALDECOXIB WARNER-LAMBERT COMPANY LLC (US) 2004-01-22 WO disclosed