SCHEMBL6259836

SCHEMBL6259836

C#C[C@@]1(O)C[C@H]2[C@@H]3CCc4cc(O)ccc4[C@H]3[C@@H](C)C[C@]2(C)C1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 8/20 0.54
ESR2 Q92731 6/20 0.54
CYP3A4 P08684 3/20 0.50
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
SHBG P04278 3/20 0.50
ABCB11 O95342 2/20 0.50
PGR P06401 2/20 0.50
AR P10275 2/20 0.50
SLC6A4 P31645 2/20 0.50
OPRM1 P35372 2/20 0.50
HTR2B P41595 2/20 0.50
SLC6A3 Q01959 2/20 0.50
SLC22A2 O15244 1/20 0.50
NR1I2 O75469 1/20 0.50
NR3C1 P04150 1/20 0.50
HTR1A P08908 1/20 0.50
ADORA3 P0DMS8 1/20 0.50
ADRB3 P13945 1/20 0.50
CYP2B6 P20813 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6257050 1.00 ESR1 (0.54) ESR1ESR2CYP3A4MEN1KMT2A
SCHEMBL6260538 0.83 ESR1 (0.66) ESR1ESR2CYP3A4MEN1KMT2A
SCHEMBL6258256 0.83 ESR1 (0.66) ESR1ESR2CYP3A4MEN1KMT2A
SCHEMBL10601350 0.81 ESR1 (0.76) ESR1ESR2CYP3A4MEN1KMT2A
SCHEMBL7642558 0.81 ESR1 (0.76) ESR1ESR2CYP3A4MEN1KMT2A
SCHEMBL11170420 0.81 ESR1 (0.76) ESR1ESR2CYP3A4MEN1KMT2A
SCHEMBL5680132 0.78 MEN1 (0.53) ESR1ESR2CYP3A4MEN1KMT2A
SCHEMBL5679659 0.78 MEN1 (0.53) ESR1ESR2CYP3A4MEN1KMT2A
SCHEMBL25863861 0.75 ESR1 (0.54) ESR1ESR2CYP3A4MEN1KMT2A
SCHEMBL25863898 0.75 ESR1 (0.54) ESR1ESR2CYP3A4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1580192-A2 16-Hydroxyestratrienes as selective estrogens Schering AG (DE) 2005-09-28 EP claimed
EP-1580192-A2 16-Hydroxyestratrienes as selective estrogens Schering AG (DE) 2005-09-28 EP disclosed