SCHEMBL6258256

SCHEMBL6258256

C#C[C@]1(O)C[C@H]2[C@@H]3CCc4cc(O)ccc4[C@H]3CC[C@]2(C)C1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 10/20 0.66
ESR2 Q92731 7/20 0.66
SHBG P04278 5/20 0.66
CYP3A4 P08684 4/20 0.66
PGR P06401 4/20 0.66
AR P10275 4/20 0.66
SLC6A4 P31645 4/20 0.66
SLC6A3 Q01959 4/20 0.66
ABCB11 O95342 3/20 0.66
HTR2B P41595 3/20 0.66
NR3C1 P04150 3/20 0.66
CYP2B6 P20813 2/20 0.66
OPRM1 P35372 2/20 0.66
SULT1A1 P50225 2/20 0.66
AOX1 Q06278 2/20 0.66
MEN1 O00255 2/20 0.66
KMT2A Q03164 2/20 0.66
SLC22A2 O15244 1/20 0.66
NR1I2 O75469 1/20 0.66
HTR1A P08908 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6260538 1.00 ESR1 (0.66) ESR1ESR2SHBGCYP3A4PGR
SCHEMBL6262096 0.88 ESR1 (0.66) ESR1ESR2SHBGCYP3A4PGR
SCHEMBL6259836 0.83 ESR1 (0.54) ESR1ESR2SHBGCYP3A4PGR
SCHEMBL6257050 0.83 ESR1 (0.54) ESR1ESR2SHBGCYP3A4PGR
SCHEMBL6257381 0.81 ESR1 (0.45) ESR1ESR2SHBGCYP3A4PGR
SCHEMBL6259610 0.81 ESR1 (0.45) ESR1ESR2SHBGCYP3A4PGR
Ethinyl Estradiol SCHEMBL4071 0.80 ESR1 (1.00) ESR1ESR2SHBGCYP3A4PGR
Ethinyl Estradiol SCHEMBL12180049 0.80 ESR1 (1.00) ESR1ESR2SHBGCYP3A4PGR
Ethinyl Estradiol SCHEMBL13575761 0.80 ESR1 (1.00) ESR1ESR2SHBGCYP3A4PGR
Ethinyl Estradiol SCHEMBL19963467 0.80 ESR1 (1.00) ESR1ESR2SHBGCYP3A4PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1580192-A2 16-Hydroxyestratrienes as selective estrogens Schering AG (DE) 2005-09-28 EP claimed
EP-1580192-A2 16-Hydroxyestratrienes as selective estrogens Schering AG (DE) 2005-09-28 EP disclosed