SCHEMBL6262863

SCHEMBL6262863

[CH2]C(c1ccc(Cl)cc1)c1ccccc1C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.47
CNR1 P21554 5/20 0.43
TSHR P16473 4/20 0.42
ALDH1A1 P00352 2/20 0.42
ACP3 P15309 1/20 0.41
P2RX7 Q99572 1/20 0.41
HIF1A Q16665 3/20 0.40
L3MBTL1 Q9Y468 3/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
MAPT P10636 2/20 0.40
ATM Q13315 2/20 0.40
LMNA P02545 2/20 0.40
MAPK1 P28482 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
KDM4E B2RXH2 1/20 0.40
NR1I2 O75469 1/20 0.40
ABCB11 O95342 1/20 0.40
NR3C1 P04150 1/20 0.40
PGR P06401 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4007134 0.85 ACP3 (0.54) CNR2TSHRALDH1A1ACP3P2RX7
SCHEMBL4189236 0.81 CNR2 (0.49) CNR2CNR1TSHRALDH1A1ACP3
SCHEMBL6260007 0.75 TSHR (0.39) CNR2CNR1TSHRALDH1A1HIF1A
SCHEMBL20547735 0.71 CNR2 (0.57) CNR2CNR1ACP3P2RX7LMNA
SCHEMBL30240014 0.71 CNR2 (0.57) CNR2CNR1ACP3P2RX7LMNA
SCHEMBL4214299 0.71 ACP3 (0.47) CNR2ALDH1A1ACP3P2RX7L3MBTL1
SCHEMBL8429801 0.71 P2RX7 (0.47) CNR2ALDH1A1ACP3P2RX7L3MBTL1
SCHEMBL3535353 0.71 TSHR (0.50) CNR1TSHRALDH1A1HIF1AL3MBTL1
SCHEMBL4710744 0.70 P2RX7 (0.40) CNR2CNR1TSHRALDH1A1P2RX7
SCHEMBL29523337 0.70 ACP3 (0.46) CNR2TSHRALDH1A1ACP3P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005077463-A2 LIGAND FOR A MONOAMINE RECEPTOR OR TRANSPORTER FOR TREATING ADDICTION OR DEPENDENCE SEPRACOR INC. (US) 2005-08-25 WO disclosed