SCHEMBL6264246

SCHEMBL6264246

OC1CCC(Nc2nc(-c3cccnc3)cn3ccnc23)CC1

nearest known ligand 0.60

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AURKA O14965 7/20 0.60
MAPK8 P45983 5/20 0.49
TYRO3 Q06418 2/20 0.47
MERTK Q12866 2/20 0.47
AXL P30530 1/20 0.47
EPHB4 P54760 1/20 0.44
FLT3 P36888 1/20 0.44
GAS6 Q14393 1/20 0.44
SYK P43405 3/20 0.43
GBA1 P04062 1/20 0.42
ADORA3 P0DMS8 1/20 0.41
TMIGD3 P0DMS9 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6280533 0.87 MAPK8 (0.50) AURKAMAPK8TYRO3MERTKEPHB4
SCHEMBL6265223 0.85 PIK3CA (0.53) AURKAMAPK8EPHB4SYK
SCHEMBL6264936 0.85 MAPK8 (0.58) AURKAMAPK8TYRO3MERTKEPHB4
SCHEMBL6270503 0.84 AURKA (0.57) AURKAMAPK8SYK
SCHEMBL6260383 0.84 SYK (0.59) AURKAMAPK8SYKADORA3TMIGD3
SCHEMBL6263352 0.84 MAPK8 (0.49) AURKAMAPK8SYKADORA3
SCHEMBL6262086 0.82 SYK (0.60) MAPK8SYK
SCHEMBL6264925 0.82 MAPK8 (0.57) MAPK8EPHB4SYKADORA3TMIGD3
SCHEMBL6264254 0.82 FYN (0.48) AURKAMAPK8EPHB4SYK
SCHEMBL6263073 0.81 RXFP1 (0.55) AURKAEPHB4SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005085252-A1 IMIDAZO ‘1,2-A’ PYRAZINE COMPOUNDS WHICH INTERACT WITH PROTEIN KINASES BIOFOCUS DISCOVERY LIMITED (GB) 2005-09-15 WO claimed