SCHEMBL6266293

SCHEMBL6266293

O=C(/C=C\c1cccnc1)NCCCCN1CCN(c2ccccc2)CC1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 12/20 0.72
DRD2 P14416 12/20 0.72
HTR1A P08908 3/20 0.67
HTR2A P28223 2/20 0.67
CYP3A4 P08684 1/20 0.58
CYP2C9 P11712 1/20 0.58
NAMPT P43490 1/20 0.58
ALOX5 P09917 1/20 0.58
HDAC3 O15379 1/20 0.56
HDAC4 P56524 1/20 0.56
HDAC1 Q13547 1/20 0.56
HDAC7 Q8WUI4 1/20 0.56
HDAC2 Q92769 1/20 0.56
HDAC10 Q969S8 1/20 0.56
HDAC11 Q96DB2 1/20 0.56
HDAC8 Q9BY41 1/20 0.56
HDAC6 Q9UBN7 1/20 0.56
HDAC9 Q9UKV0 1/20 0.56
HDAC5 Q9UQL6 1/20 0.56
DRD4 P21917 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6266296 1.00 DRD3 (0.72) DRD3DRD2HTR1AHTR2ACYP3A4
SCHEMBL82842 0.87 DRD2 (0.73) DRD3DRD2HTR1ACYP3A4CYP2C9
SCHEMBL3074410 0.87 DRD2 (0.73) DRD3DRD2HTR1ACYP3A4CYP2C9
SCHEMBL3076885 0.86 NAMPT (0.74) DRD3DRD2HTR1AHTR2ACYP3A4
SCHEMBL82431 0.86 NAMPT (0.74) DRD3DRD2HTR1AHTR2ACYP3A4
SCHEMBL3086811 0.86 DRD2 (0.72) DRD3DRD2HTR1ACYP3A4CYP2C9
SCHEMBL82104 0.86 DRD2 (0.72) DRD3DRD2HTR1ACYP3A4CYP2C9
SCHEMBL82749 0.86 DRD2 (0.72) DRD3DRD2HTR1ACYP3A4CYP2C9
SCHEMBL3073890 0.86 DRD2 (0.72) DRD3DRD2HTR1ACYP3A4CYP2C9
SCHEMBL13276712 0.86 DRD2 (0.61) DRD3DRD2CYP3A4CYP2C9NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1079832-B1 USE OF VITAMIN PP COMPOUNDS KLINGE CO CHEM PHARM FAB (DE) 2005-11-30 EP claimed